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6-(2,5-dimethylfuran-3-yl)-7-methyl-2-(piperidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(2S,3S)-3-methyl-2-({[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]carbamoyl}amino)pentanamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(pyridin-3-ylmethyl)acetamide
1-(1H-indole-6-carbonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
4-(6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-4-oxobutanamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
1-[benzyl(methyl)sulfamoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}-8-fluoro-1,4-dihydroquinolin-4-one
({1-[(1-hexylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)(methyl)amine
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-methyl-3-(morpholin-4-yl)propan-1-one
5-(2,3-dimethylphenyl)-1,2-dihydropyrimidin-2-one
2-butoxy-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)acetamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-[2-(3-methoxyphenyl)-1-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(3,3,4,4-tetrafluorobutyl)morpholine
1-methyl-N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-pyrazole-5-carboxamide
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
2-[(3-methyl-1-phenyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-benzyl-4-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
4-(4-methyl-1H-pyrazol-1-yl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidine-4-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-(2-fluoroethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-chloro-2-methoxy-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
4-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
(3aR,7aS)-2-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-[2-(pyridin-2-yl)ethyl]piperidine-1-carboxamide
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]azocane
N-cyclopentyl-1-methyl-5-[2-(1,3-thiazol-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-3-yl)acetamide
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-{[4-(methylsulfanyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,4-diazepan-2-one
1-(4-hydroxypiperidin-1-yl)-3-[5-(pent-2-yn-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propan-1-one
1-[(2-chlorophenyl)methyl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-ethyl-8-[(3-hydroxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methylthiophen-2-yl)methyl]amine
4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-1,4-oxazepan-6-ol
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(1-methyl-1H-imidazol-2-yl)benzamide
3-{[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]methyl}-N,N-dimethylpyridin-2-amine
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[4-(hydroxymethyl)phenyl]ethan-1-one
2-{[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
1-[3-(4-fluorophenyl)phenyl]-N-[2-(1H-imidazol-4-yl)ethyl]piperidin-4-amine
1-butanoyl-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
2-({4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}methyl)pyridine
N-benzyl-2-{2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}propanamide
3-benzyl-1-methyl-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrazole-4-carboxamide
4-methyl-7-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}-2H-chromen-2-one
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide