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3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-(4-ethylpiperazin-1-yl)-N-(1,2-oxazol-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-[2-(4-propylmorpholin-2-yl)ethyl]pyrazolo[1,5-a]pyridine-2-carboxamide
2-(2-aminopyridine-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{4-[7-(6,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidin-1-yl}ethan-1-one
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrrolidine-1-sulfonamide
6-(methoxymethyl)-1-methyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1H-pyrazolo[3,4-d]pyrimidine
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}propan-1-one
4-(morpholin-4-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
2,4-dimethyl-7-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
8-(1-methoxypropan-2-yl)-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-N-(4-cyano-2-fluorophenyl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carboxamide
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-N,N-diethylpyrrolidin-3-amine
1'-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{3-[(cyclopentylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
(2S,4R)-1-benzyl-N-[2-(dimethylamino)ethyl]-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
1-[(3S)-3-ethylmorpholin-4-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-(3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2-methylphenyl)furan-2-carboxamide
7-[(4-phenylpiperazin-1-yl)methyl]-4-(1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(azepan-1-yl)-1-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
3-(3,4-dimethoxybenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
1-[3-({3-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-cyclohexyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(methylsulfanyl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
{[2-(2-methoxyphenyl)-6-methylquinolin-3-yl]methyl}(2-methylpropyl)amine
2,2-dimethyl-N-(1-{1-[1-(4-methylphenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
(3R,4S)-N,N-dimethyl-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(propan-2-yl)pyrrolidin-3-amine
(5S,9aS,9bS)-5-[2-(4-chlorophenyl)pyrimidin-5-yl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(2,4-diethoxy-3-methylphenyl)methyl]piperidine-4-carbonitrile
(1R,5R)-3-benzoyl-6-[(2,3,4-trifluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(2R,3S,6R)-3-(3-methoxyphenyl)-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
1-methyl-4-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}piperazine-2-carboxylic acid
methyl 1-[(3R,5S)-1-(adamantan-2-yl)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridazine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-2-(methylamino)pyrimidine-5-carboxamide
2-(3-chlorophenyl)-4-[4-(cyclohexylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[5-(1-benzoylpiperidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
2-[methyl(pyridin-3-ylmethyl)amino]-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
8-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(5-methylthiophen-2-yl)methyl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
(2S,4S)-4-amino-1-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)pyrrolidine-2-carboxylic acid
N-[(2S)-2-hydroxypropyl]-4-{[2-(2-oxopyrrolidin-1-yl)ethyl]sulfamoyl}benzamide
3-methoxy-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
(4aS,7aR)-1-(2-hydroxy-5-methylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}imidazolidine-2,4-dione
methyl 4-{[4-(quinazolin-4-yl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate