Sulpiride

• 产品号: Bio-0717
• CAS号: 15676-16-1
• 分子式: C15H23N3O4S
• 分子量: 341.42582

产品别名

• 标题: Sulpiride
• IUPAC标准名: N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-5-sulfamoylbenzamide
• IUPAC传统名: N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-5-sulfamoylbenzamide
• 别名: Milsulvan; Mirbanil; Dogmatil; Dogmatyl; Eglonyl

产品登记号

• CAS号: 15676-16-1

产品性质

• 应用领域: Low acute toxicity
• 应用领域: Antidepressant
• 应用领域: Digestive aid
• 应用领域: Antianxiety drug
• 应用领域: Non-sedative major antipsychotic agent
• 应用领域: Migraine therapeutic
• 生物活性机理: Dopamine D2-receptor antagonist
• 生物活性机理: In contrast to most other neuroleptics which block both dopamine D1 and D2 receptors, Sulpiride is more selective and acts primarily as a dopamine D2 antagonist
• 生物活性机理: Sulpiride appears to lack effects on norepinephrine, acetylcholine, serotonin, histamine, or gamma-aminobutyric acid (GABA) receptors

参考文献

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