Sulfadimidine

• 产品号: Bio-0716
• CAS号: 57-68-1
• 分子式: C12H14N4O2S
• 分子量: 278.33016

产品别名

• 标题: Sulfadimidine
• IUPAC标准名: 4-amino-N-(4,6-dimethylpyrimidin-2-yl)benzene-1-sulfonamide
• IUPAC传统名: 4-amino-N-(4,6-dimethylpyrimidin-2-yl)benzene-1-sulfonamide
• 别名: Sulphamezathine; Sulfadimesine; Sulfamethazine; Sulfodimezine; Sulphadimidine; Sulfadimethylpyrimidine; Sulfadimezine; Superseptil; Sulphamethazine; Sulfadimerazine

产品登记号

• CAS号: 57-68-1

产品性质

• 应用领域: Antiseptic
• 应用领域: Widely-used, short acting sulfonamide, used in treatment of systemic and urinary tract infections
• 应用领域: Low acute toxicity
• 生物活性机理: Sulfonamides, being structural analogues of para-aminobenzoic acid (PABA), competitively inhibit the incorporation of PABA into dihydropteric acid, the precursor of folic acid.
• 生物活性机理: Subsequent reduction in the level of folic acid reduced the production of nucleic acids in sensitive bacteria.
• 生物活性机理: Folate-antagonist
• 生物活性机理: Dihydrofolate-reductase inhibitor
• 生物活性机理: Dihydrofolate-synthesis inhibitor

参考文献

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