Δ4-Tibolone

• 产品号: T437505
• CAS号: 1162-60-3
• 分子式: C21H28O2
• 分子量: 312.44582
• 保 存: -20°C Freezer

产品别名

• 标题: Δ4-Tibolone
• IUPAC标准名: (1S,2R,9R,10R,11S,14R,15S)-14-ethynyl-14-hydroxy-9,15-dimethyltetracyclo[8.7.0.0^2,^7.0^1^1,^1^5]heptadec-6-en-5-one
• IUPAC传统名: (1S,2R,9R,10R,11S,14R,15S)-14-ethynyl-14-hydroxy-9,15-dimethyltetracyclo[8.7.0.0^2,^7.0^1^1,^1^5]heptadec-6-en-5-one
• 别名: Org-OM 38; NSC 142228; 7α-Methylnorethindrone; 17α-Ethynyl-17-hydroxy-7α-methyl-4-estren-3-one; (7α,17α)-17-Hydroxy-7-methyl-19-norpregn-4-en-20-yn-3-one

产品登记号

• CAS号: 1162-60-3

产品性质

• 外观: Off-White Solid
• 熔点: 203-205°C
• 溶解度: Dichloromethane
• 溶解度: Ethyl Acetate
• 溶解度: Methanol
• 保存条件: -20°C Freezer

产品详细信息

详细说明 (English)

A metabolite of Tibolone. A synthetic steroid with weak estrogenic, androgenic and progestogenic activity. A pharamceutical used in the treatment of menopausal syndrome.

参考文献

• Landgren, M., et al.: Maturitas, 50, 222 (2001)
• Wang, M., et al.: Steroids, 71, 343 (2001)
• Verheul, H., et al.: Drug Metab. Dispos., 35, 1105 (2001)
• Clarkson, T., et al.: J. Clin. Endocrinol. Metab., 86, 5396 (2001)