Tapentadol-d5 Hydrochloride

• 产品号: T007202
• 分子式: C14H24ClNO
• 分子量: 257.79946
• 保 存: -20°C Freezer, Under Inert Atmosphere

产品别名

• 标题: Tapentadol-d5 Hydrochloride
• IUPAC标准名: 3-[(2R,3R)-1-(dimethylamino)-2-methyl(4,4,5,5,5-^2H₅)pentan-3-yl]phenol hydrochloride
• IUPAC传统名: 3-[(2R,3R)-1-(dimethylamino)-2-methyl(4,4,5,5,5-^2H₅)pentan-3-yl]phenol hydrochloride
• 别名: 3-[(1R,2R)-3-(Dimethylamino)-1-(ethyl-d5)-2-methylpropyl]phenol Hydrochloride

产品性质

• 外观: Off-White Solid
• 熔点: 188-206°C
• 溶解度: Methanol
• 保存条件: -20°C Freezer, Under Inert Atmosphere

产品详细信息

详细说明 (English)

A novel, centrally acting oral analgesic with a dual mode of action that has demonstrated efficacy in preclinical and clinical models of pain relief.

参考文献

• Boxenbaum, H., et al.: J. Pharm. Sci., 2, 47 (1999)
• Boase, S., et al.: Br. J. Clin. Pharmacol., 54, 493 (1999)
• Armstrong, S., et al.: Psychosomatics, 44, 515 (1999)
• Bjornsson, T., et al.: Drug Metab. Dispos., 31, 815 ( 2003),