Rupatadine Fumarate

• 产品号: R701650
• CAS号: 182349-12-8
• 分子式: C30H30ClN3O4
• 分子量: 532.0299
• 保 存: Refrigerator

产品别名

• 标题: Rupatadine Fumarate
• IUPAC标准名: (2E)-but-2-enedioic acid; 13-chloro-2-{1-[(5-methylpyridin-3-yl)methyl]piperidin-4-ylidene}-4-azatricyclo[9.4.0.0^3,^8]pentadeca-1(11),3(8),4,6,12,14-hexaene
• IUPAC传统名: 13-chloro-2-{1-[(5-methylpyridin-3-yl)methyl]piperidin-4-ylidene}-4-azatricyclo[9.4.0.0^3,^8]pentadeca-1(11),3(8),4,6,12,14-hexaene; fumaric acid
• 别名: 8-Chloro-6,11-dihydro-11-[1-[(5-methyl-3-pyridinyl)methyl]-4-piperidinylidene]-5H-benzo[5,6]cyclohepta[1,2-b]pyridine (2E)-2-Butenedioate; Rupafin

产品登记号

• CAS号: 182349-12-8

产品性质

• 外观: White Solid
• 熔点: 196-198°C
• 溶解度: Methanol
• 保存条件: Refrigerator

产品详细信息

详细说明 (English)

Rupatadine is a dual antagonist of histamine H1 and platelet-activating factor receptors. Rupatadine is used as an antihistaminic.

参考文献

• Merlos, M., et al.: J. Pharmacol. Exp. Ther., 280, 114 (1997)
• Guadano, E.M., et al.: Allergy, 59, 766 (1997)