Raloxifene-d4 4'-Glucuronide

• 产品号: R100022
• 分子式: C34H35NO10S
• 分子量: 649.7074
• 保 存: -20°C Freezer

产品别名

• 标题: Raloxifene-d4 4'-Glucuronide
• IUPAC标准名: (2R,3R,4R,5S,6R)-3,4,5-trihydroxy-6-[4-(6-hydroxy-3-{4-[2-(piperidin-1-yl)(^2H₄)ethoxy]benzoyl}-1-benzothiophen-2-yl)phenoxy]oxane-2-carboxylic acid
• IUPAC传统名: (2R,3R,4R,5S,6R)-3,4,5-trihydroxy-6-[4-(6-hydroxy-3-{4-[2-(piperidin-1-yl)(^2H₄)ethoxy]benzoyl}-1-benzothiophen-2-yl)phenoxy]oxane-2-carboxylic acid
• 别名: 4-[6-Hydroxy-3-[4-[2-(1-piperidinyl)ethoxy-d4]benzoyl]benzo[b]thien-2-yl]phenyl-β-D-glucopyranosiduronic Acid

产品性质

• 外观: Yellow Solid
• 熔点: 207-212°C (dec.)
• 溶解度: DMF
• 溶解度: DMSO
• 溶解度: Hot Methanol
• 保存条件: -20°C Freezer

产品详细信息

详细说明 (English)

A labelled metabolite of Raloxifene, a nonsteroidal estrogen receptor mixed agonist/antagonist.

参考文献

• Dodge, J., et al.: Bioorg. Med. Chem. Lett., 7, 993 (1997)
• Jeong, E., et al.: Drug Metab. Dispos., 33, 785 (1997)
• Trontelj, J., et al.: Pharmacol. Res., 52, 334 (1997)
• Oswald, S., et al.: Clin. Pharmacol. Ther., 79 206 (1997)