5-Pyrimidineboronic Acid Pinacol Ester

• 产品号: P997260
• CAS号: 321724-19-0
• 分子式: C10H15BN2O2
• 分子量: 206.0493

产品别名

• 标题: 5-Pyrimidineboronic Acid Pinacol Ester
• IUPAC标准名: 5-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidine
• IUPAC传统名: 5-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidine
• 别名: 5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidine; Pyrimidyl-5-boronic acid pinacolate

产品登记号

• CAS号: 321724-19-0

产品详细信息

详细说明 (English)

2-Methoxyphenylborornic Acid Pinacol Ester is used in the preparation of indole derivatives as selective inhibitors of all three members of the Pim kinase family. It is also used to prepare inhibitors of TGF-β1 and activin A signalling.

参考文献

• Nishiguchi, G.A. et al.: Bioorg. Med. Chem. Lett., 21, 6366 (2011)
• Ciayadi, R. et al.: Bioorg. Med. Chem. Lett., 21, 5642 (2011)