Oripavine-d3

• 产品号: O675002
• 分子式: C18H19NO3
• 分子量: 297.34836
• 保 存: Controlled Substance, -20°C Freezer

产品别名

• 标题: Oripavine-d3
• IUPAC标准名: (1S,5S,13R)-14-methoxy-4-(^2H₃)methyl-12-oxa-4-azapentacyclo[9.6.1.0^1,^1^3.0^5,^1^7.0^7,^1^8]octadeca-7(18),8,10,14,16-pentaen-10-ol
• IUPAC传统名: (1S,5S,13R)-14-methoxy-4-(^2H₃)methyl-12-oxa-4-azapentacyclo[9.6.1.0^1,^1^3.0^5,^1^7.0^7,^1^8]octadeca-7(18),8,10,14,16-pentaen-10-ol
• 别名: 3-O-Demethylthebaine; (5α)-6,7,8,14-Tetradehydro-4,5-epoxy-6-methoxy-17-methylmorphinan-3-ol

产品性质

• 外观: Gray Solid
• 熔点: 183-187°C (dec.)
• 溶解度: Chloroform
• 溶解度: Methanol
• 保存条件: Controlled Substance, -20°C Freezer

产品详细信息

详细说明 (English)

The major metabolite of Thebaine. Oripavine possesses an analgesic potency comparable to Morphine; it is not clinically useful due to severe toxicity and low therapeutic index. An opiate.

参考文献

• Barber, R., et al.: J. Med. Chem., 18, 1074 (1975)
• Yamazoe, Y., et al.: J. Pharmacol., 31, 433 (1975)