6-Methyl Pergolide

• 产品号: M326070
• CAS号: 57202-76-3
• 分子式: C17H22N2S
• 分子量: 286.43498
• 保 存: Refrigerator

产品别名

• 标题: 6-Methyl Pergolide
• IUPAC标准名: (2R,4R,7R)-6-methyl-4-[(methylsulfanyl)methyl]-6,11-diazatetracyclo[7.6.1.0^2,^7.0^1^2,^1^6]hexadeca-1(16),9,12,14-tetraene
• IUPAC传统名: (2R,4R,7R)-6-methyl-4-[(methylsulfanyl)methyl]-6,11-diazatetracyclo[7.6.1.0^2,^7.0^1^2,^1^6]hexadeca-1(16),9,12,14-tetraene
• 别名: (8β)-6-Methyl-8-[(methylthio)methyl]ergoline; LY 116467; LY 062

产品登记号

• CAS号: 57202-76-3

产品性质

• 外观: White to Off-White Solid
• 熔点: >256°C (dec.)
• 溶解度: Chloroform
• 溶解度: Dichloromethane
• 溶解度: Dimethylformamide
• 溶解度: Methanol
• 保存条件: Refrigerator

产品详细信息

详细说明 (English)

Potent antagonist of 5-HT2A and 5-HT2B receptors on porcine cardiac valves, it also activates brain dopaminergic receptors and lowers cranial DOPAC levels in rats.

参考文献

• Fuller, R.W., et al.: Neuroendocrinol., 36, 285 (1983)
• Goernemann, T., et al.: J. Pharmacol. Exp. Ther., 324, 1136 (1983)