CGS-9343B

• 产品号: C1619
• CAS号: 109826-27-9
• 分子式: C30H32N4O6
• 分子量: 544.59828
• 纯 度: ≥98% (HPLC)

产品别名

• 标题: CGS-9343B
• IUPAC标准名: 1-[1-({7-methyl-8-oxa-2-azatricyclo[8.4.0.0^2,^6]tetradeca-1(14),3,5,10,12-pentaen-7-yl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one; but-2-enedioic acid
• IUPAC传统名: 1-[1-({7-methyl-8-oxa-2-azatricyclo[8.4.0.0^2,^6]tetradeca-1(14),3,5,10,12-pentaen-7-yl}methyl)piperidin-4-yl]-3H-1,3-benzodiazol-2-one; butenedioic acid
• 别名: Zaldaride maleate; CGS9343B; KW-5617; 1,3-Dihydro-1-[1-[(4-methyl-4H,6H-pyrrolo[1,2-a][4,1]- benzoxazepin-4-yl)methyl]-4-piperidinyl]-2H-benzimidazol-2-one maleate

产品登记号

• MDL号: MFCD04113002
• CAS号: 109826-27-9

产品性质

• Empirical Formula (Hill Notation): C26H28N4O2 · C4H4O4
• 纯度: ≥98% (HPLC)
• 外观: white to off-white powder
• 溶解度: DMSO: >10 mg/mL
• 保存温度: 2-8°C
• 德国WGK号: 3

产品详细信息

详细说明 (English)

Biochem/physiol Actions
CGS-9343B is a selective calmodulin antagonist with minimal protein kinase C or antidopaminergic activity. CGS-9343B is a potent inhibitor of calmodulin-activated (Type I) phosphodiesterase activity with IC50 in the nanomolar range.

详细说明 (简体中文)

Biochem/physiol Actions
CGS-9343B is a selective calmodulin antagonist with minimal protein kinase C or antidopaminergic activity. CGS-9343B is a potent inhibitor of calmodulin-activated (Type I) phosphodiesterase activity with IC50 in the nanomolar range.