[β-Mercapto-β,β-cyclopentamethylenepropionyl1, O-Et-Tyr2, Val4, Arg8]-Vasopressin

• 产品号: V4253
• CAS号: 77453-01-1
• 分子式: C53H77N13O11S2
• 分子量: 1136.38898
• 纯 度: ≥97% (HPLC)

产品别名

• 标题: [β-Mercapto-β,β-cyclopentamethylenepropionyl1, O-Et-Tyr2, Val4, Arg8]-Vasopressin
• IUPAC标准名: (2S)-2-{[(2S)-1-[(10R,13S,16S,19S,22S)-19-benzyl-13-(carbamoylmethyl)-22-[(4-ethoxyphenyl)methyl]-12,15,18,21,24-pentaoxo-16-(propan-2-yl)-7,8-dithia-11,14,17,20,23-pentaazaspiro[5.19]pentacosane-10-carbonyl]pyrrolidin-2-yl]formamido}-5-carbamimidamido-N-(carbamoylmethyl)pentanamide
• IUPAC传统名: (2S)-2-{[(2S)-1-[(10R,13S,16S,19S,22S)-19-benzyl-13-(carbamoylmethyl)-22-[(4-ethoxyphenyl)methyl]-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaazaspiro[5.19]pentacosane-10-carbonyl]pyrrolidin-2-yl]formamido}-5-carbamimidamido-N-(carbamoylmethyl)pentanamide

产品登记号

• MDL号: MFCD00076752
• CAS号: 77453-01-1

产品性质

• 纯度: ≥97% (HPLC)
• 相关基因信息: human ... AVPR1A(552), AVPR2(554), OXT(5020), OXTR(5021)mouse ... AVPR1A(54140), AVPR2(12000)rat ... AVPR1A(25107), AVPR2(25108), OXT(18429), OXTR(18430)
• GHS警示词: Warning
• GHS危险声明: H332
• 欧盟危险性物质标志: 有害性(Harmful) (Xn)
• 个人保护装置: dust mask type N95 (US), Eyeshields, Gloves
• 危险公开号: 20
• 安全公开号: 36
• 保存温度: -20°C
• 德国WGK号: 3

产品详细信息

详细说明 (English)

Amino Acid Sequence
(1-Mercaptocyclohexyl)acetyl-Tyr(O-Ethyl)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 [Disulfide Bridge: 1-6]
Biochem/physiol Actions
Potent V1a and V2 vasopressin receptor and oxytocin receptor antagonist.