Ritanserin

• 产品号: R103
• CAS号: 87051-43-2
• 分子式: C27H25F2N3OS
• 分子量: 477.5687064

产品别名

• 标题: Ritanserin
• IUPAC标准名: 6-(2-{4-[bis(4-fluorophenyl)methylidene]piperidin-1-yl}ethyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
• IUPAC传统名: ritanserin
• 别名: 6-[2-[4-(bis(4-Fluorophenyl)methylene]-1-piperidinyl]ethyl]-7-methyl-5H-thiazolo[3,2-a]pyrimidin-5-one

产品登记号

• MDL号: MFCD00069341
• CAS号: 87051-43-2
• PubChem SID: 24278117

产品性质

• 相关基因信息: human ... HTR2A(3356)rat ... Adra1a(29412), Drd2(24318), Htr1a(24473), Htr2a(29595), Htr7(65032)
• 外观: white powder
• 溶解度: methanol: >10 mg/mL
• 溶解度: DMSO: >10.1 mg/mL
• 溶解度: 2-hydroxypropyl-β-cyclodextrin: insoluble
• 溶解度: H2O: insoluble
• 溶解度: dilute aqueous base: insoluble
• GHS警示词: Warning
• GHS危险声明: H315-H319-H335
• 欧盟危险性物质标志: 刺激性(Irritant) (Xi)
• 个人保护装置: dust mask type N95 (US), Eyeshields, Gloves
• GHS警示性声明: P261-P305 + P351 + P338
• 危险公开号: 36/37/38
• 安全公开号: 22-26-36
• 德国WGK号: 3

产品详细信息

详细说明 (English)

Biochem/physiol Actions
Potent 5-HT2A serotonin receptor antagonist/inverse agonist that crosses the blood-brain barrier.
Other Notes
Tandem Mass Spectrometry data independently generated by Scripps Center for Metabolomics is available to view or download in PDF. R103.pdf Tested metabolites are featured on Scripps Center for Metabolomics METLIN Metabolite Database. To learn more, visit sigma.com/metlin.