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[3-(3-methylbut-2-en-1-yl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl]methanol
5-(methoxymethyl)-3-{[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
7-fluoro-N-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
5-{1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl}-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-[1-(2-fluorophenyl)piperidin-4-yl]-4-(pyridin-3-yl)pyrimidin-2-amine
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylic acid
5-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzothiadiazole
(4aS,7aR)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(2,3-dihydro-1H-inden-1-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]-1-(1,2-oxazole-5-carbonyl)piperidine
4-(1-benzofuran-5-carbonyl)-1-(3,5-dimethylphenyl)piperazin-2-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidine
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
[3-(1H-imidazol-1-yl)propyl](2-phenylethyl)(pyridin-3-ylmethyl)amine
4-{2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-2-one
4-{1-[(5-methylpyrazin-2-yl)methyl]-1H-imidazol-2-yl}-2-(propan-2-yl)pyrimidine
4-[5-(5-butylpyridine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]morpholine
N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[1-(pyridin-2-yl)ethyl]butanamide
1-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[(2,2-dimethyloxan-4-yl)methyl]-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
N-[1-(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-phenylpropanamide
3-(4-chlorophenyl)-2-{[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}propan-1-ol
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2,2-dimethyl-N-(pyridin-4-ylmethyl)oxane-4-carboxamide
2-({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethan-1-ol
3-[3-(1H-1,3-benzodiazol-2-yl)azetidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
(3R,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
3,5-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)furan-2-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
ethyl 1-(pyridine-2-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(4-phenyloxan-4-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
1-(1-benzylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
4-[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]pyrimidine
4-(1-{[5-(furan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrrolidin-3-yl)morpholine
(1S,5R)-3-(pyrazine-2-carbonyl)-6-(thiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(2,6-dimethylpyridin-3-yl)-N-[2-(4-methylpiperazin-1-yl)propyl]pyrimidin-2-amine
2-(4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazin-1-yl)pyrimidine
5-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
methyl 2-{[4-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]sulfonyl}benzoate
methyl 3-[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]benzoate
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-fluoro-N-(propan-2-yl)-5-sulfamoylbenzamide
(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-methoxy-3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(5-methyl-1H-pyrazole-3-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
4-{4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-1-yl}butan-1-ol
{9-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-3-(3-methylbut-2-en-1-yl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
2-[4-(4-methoxyphenoxy)piperidin-1-yl]quinoline