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N-[2-(pyrrolidine-1-sulfonyl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(ethylsulfanyl)ethyl]-4-(piperazine-1-sulfonyl)benzamide
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
1-phenyl-4-[1-(thiophene-3-sulfonyl)piperidin-3-yl]piperazine
2-[1-(2-methylpropyl)-4-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(methylsulfamoyl)ethyl]propanamide
2-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}-3-methylquinoxaline
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
1-(3,5-difluorophenyl)-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(2-{[(4-cyclopentylpyrimidin-2-yl)amino]methyl}morpholin-4-yl)ethan-1-one
5-(2-chloro-4-fluorophenyl)-3-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
6-[3-(azepan-1-yl)-2-hydroxypropyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1-methyl-1H-indole
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-N-(2-chlorophenyl)propanamide
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-2-methoxyphenol
6-fluoro-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
(2S,4S)-4-amino-N-methyl-1-{[4-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
2-methyl-5-{[3-(4-phenylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}pyridine
2-{1-methyl-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-2-yl}ethan-1-ol
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
3-[3-(furan-2-yl)-5-(5-propylthiophen-3-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
1-[(3-methoxyphenyl)methyl]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
1-[3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-6-methylquinolin-2-yl]piperidin-3-ol
5-butyl-4-(1H-pyrrole-2-carbonyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)piperazin-2-one
3-(1-benzoylpiperidin-4-yl)-1-(4-benzylpiperidin-1-yl)propan-1-one
6-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]pyridine-3-carboxamide
1-{4-[2-(3,4-dimethoxyphenyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-methoxyethan-1-one
N-[(5-chlorothiophen-2-yl)methyl]-3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-[2-(3-fluorophenyl)ethyl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-6-(3-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(1-ethyl-1H-pyrazol-4-yl)-1-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}urea
6-{[1-(4-methoxyphenyl)piperidin-4-yl]amino}-2-methylheptan-2-ol
2-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
5-[(2-ethyl-1H-imidazol-1-yl)methyl]-3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole
2-(2-chloro-4-fluorophenyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(morpholin-3-yl)-N-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}acetamide
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[2-(2-fluorophenyl)ethyl]acetamide
2-(4-methoxyphenyl)-1-(7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-(cyclopent-3-ene-1-carbonyl)-4-[(2-methyl-1H-imidazol-4-yl)methyl]-1,4-diazepan-6-ol
1-[(2-methoxyphenyl)methyl]-4-{1H-pyrrolo[2,3-c]pyridin-5-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
8-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)ethan-1-one
N-cyclopropyl-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}-2-(trifluoromethyl)benzamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-(4-{[2-(1H-imidazol-4-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1H-indole-6-carboxamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
4-[(6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-3-yl)methyl]morpholine
5-{1-[(3-methoxyphenyl)methyl]pyrrolidin-2-yl}-N-(1H-pyrazol-3-yl)thiophene-2-carboxamide
N-(6-phenoxypyridin-3-yl)-1-(pyridine-2-carbonyl)piperidine-4-carboxamide