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5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
3-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1H-indole
2-{[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
N-[5-({4-[4-(3-methylbutyl)-2,5-dioxoimidazolidin-4-yl]piperidin-1-yl}methyl)thiophen-2-yl]acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(1,3-thiazol-2-ylmethyl)piperazine
[(1-ethyl-1H-imidazol-2-yl)methyl][(2-ethylpyrimidin-4-yl)methyl]methylamine
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-{[(2-chlorophenyl)methyl]sulfanyl}ethan-1-one
methyl[(1-propyl-1H-imidazol-2-yl)methyl]{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-(5-aminopentyl)-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
(1R,2R,4R)-N-[(6-chloropyridin-3-yl)methyl]-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-fluorobenzene-1-sulfonamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
3-(1H-imidazol-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one
1,5-dimethyl-4-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
2-(2-ethylpyrimidin-5-yl)-7-fluoro-N-methyl-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
(2E)-1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-3-(pyridin-2-yl)prop-2-en-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,1-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethan-1-amine
(1S,5R)-6-{[2-(methylsulfanyl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(2S,6S)-4-(2-methyl-6-propylpyrimidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(1R)-1-(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-amine
1-(2H-1,3-benzodioxol-5-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
(4aS,8aR)-6-(3-ethyl-1H-pyrazole-5-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-methanesulfonyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrrolidine-2-carboxamide
(1-{[methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}cyclopentyl)methanol
5-{2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-1H-1,2,3,4-tetrazole
3-methyl-7-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-{[4-(4-chlorophenoxy)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-(2-fluoro-4-methoxyphenyl)-5-methyl-4-[(2-propyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-amino-6-(1-ethyl-1H-indol-3-yl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
(4-{[4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-{2-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
7-[(3,4-difluorophenyl)methyl]-2-[(2-methylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decane
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
(5S,9aS,9bS)-5-(3-hydroxyphenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-(2-methylbenzenesulfonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-methyl-6-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzoxazole
methyl 7-oxo-9-(3-phenylpropoxy)-3-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[1-(1,3-oxazole-5-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
ethyl 4-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)piperidine-1-carboxylate
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
(3-methylbut-2-en-1-yl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
9-(3-fluoropyridine-2-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-tert-butyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
methyl 2-[(1-{4-[2-(3-fluorophenyl)acetamido]phenyl}piperidin-4-yl)amino]-4-(methylsulfanyl)butanoate