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{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
6-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2-(2-methoxyethyl)-1,3-benzoxazole
N-[2-(3-fluoro-4-methoxybenzoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
4-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-1,2-dihydrophthalazin-1-one
3-methyl-5-(1-{4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}propyl)-1,2,4-oxadiazole
2-ethyl-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[4.5]decan-3-one
1-[4-(2-{[cyclohexyl(prop-2-yn-1-yl)amino]methyl}quinazolin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
4-benzyl-3-(1-cyclopropanecarbonylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-ethyl-2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
3-[(2,4-dimethylphenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[2-(pyridin-2-yl)ethyl]quinoline-4-carboxamide
4-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperazine-2-carboxylic acid
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(3-hydroxypiperidin-1-yl)pyridine-3-carboxamide
5-{4-[(4-benzoylpiperazin-1-yl)methyl]phenyl}pyrimidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,2,7,8-tetramethylquinoline-4-carboxamide
3-ethyl-1-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]urea
4-chloro-N-[3-(oxolan-3-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(5-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
2-(1-{[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2,4-dimethyl-1,3-thiazole
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(pyridin-3-yl)ethan-1-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
5-[(3-phenyl-1H-pyrazol-1-yl)methyl]-3-propyl-1,2,4-oxadiazole
1-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
[1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
8-({4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methoxy)quinoline
(2R,4S)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-hydroxypiperidine-2-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-cyclopropaneamido-4-methylbenzamide
5-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-8-methylquinoline
2-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]pyridine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(quinolin-4-ylmethyl)amine
4-fluoro-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
(3S,4R)-N,N-dimethyl-1-{[2-(methylsulfanyl)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-amine
1-[(4-fluorophenyl)methyl]-5-(4-methoxy-2-methylbenzoyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-methoxypyridine-3-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(1R,2S)-2-propylcyclopropanecarbonyl]piperidine-4-carboxamide
1-(5-{[(3-cyclopentylpropyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
3-[(dimethylamino)methyl]-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}pyrrolidin-3-ol
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
2,6-dimethyl-N-propyl-N-(thiophen-3-ylmethyl)pyridine-4-carboxamide
1-{2-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrrolidin-1-yl}ethan-1-one
4-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-5-ethylpyrimidin-2-amine
N-ethyl-4-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-amine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)(naphthalen-1-ylmethyl)amine
6-methoxy-2-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline