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(2R)-2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-phenylpropan-1-ol
N-[2-(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclohexanecarboxamide
N-(3-ethoxy-2-hydroxypropyl)-2,7,8-trimethylquinoline-4-carboxamide
1-cyclohexyl-4-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazine
1-{3-oxo-3-[2-(2-phenylethyl)morpholin-4-yl]propyl}pyrrolidin-2-one
N-[4-fluoro-3-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]carbamoyl}amino)phenyl]propanamide
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[4-(pyridin-2-yl)phenyl]methyl}amine
2-(2-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
5-cyclopentanecarbonyl-2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-cyclopropanecarbonyl-1'-(4-ethenylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)-N-[2-(methylsulfanyl)phenyl]piperidine-1-carboxamide
4-methyl-2-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-(2-{7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
1-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-ol
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(4-ethylpiperazin-1-yl)acetamide
(3aR,6aR)-2-(4-cyclobutyl-6-methylpyrimidin-2-yl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-(furan-2-carbonyl)-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,4-diazepane
2-{[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amino}-N-methylethane-1-sulfonamide
9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N4-methyl-6-(morpholin-4-yl)pyrimidine-2,4-diamine
6-(4-chlorophenyl)-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
dimethyl(2-{2-[1-(2-methylquinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
(4aS,8aR)-1-(2-aminoethyl)-6-(5-fluoro-1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-{[4-(4-chloro-3-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}cyclopentane-1-carboxylic acid
1-(furan-2-carbonyl)-4-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
2-(dimethylamino)-4-methyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}pyrimidine-5-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-(2-phenylpropyl)piperidine-4-carboxamide
methyl 3-[2-oxo-6-(pyridin-4-ylmethoxy)-4-[2-(thiophen-2-yl)acetyl]-1,4-diazepan-1-yl]propanoate
2-[4-(3-methylbut-2-en-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-phenoxypropan-2-ol
4-(2-cyclopentylethyl)-1-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole
3-ethyl-8-(4-methyl-2-phenylpyrimidine-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{2-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
4-(4-fluorophenyl)-2-[1-(oxolan-3-ylmethyl)-1H-imidazol-2-yl]-1,3-thiazole
5-[(6-methylpyridin-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-[5-(2,3-dimethyl-1H-indole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-methyl-2-(3-{3-[2-(methylsulfanyl)phenyl]phenyl}-1H-pyrazol-1-yl)acetamide
9-[2-(3-fluoro-4-phenylphenyl)propanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
4-{1-[(2,6-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
N-phenyl-5-(3-propyl-1,2,4-oxadiazol-5-yl)pyrimidin-2-amine
N-[(2R,3R)-1'-(4-fluorobenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-{1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]piperidin-3-yl}-3-methylbutan-1-one
N-[2-(3,5-dimethylphenoxy)ethyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methylpropanamide
5-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,3,4-oxadiazol-2-amine
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazine
2,6-difluoro-N-({7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine