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N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
N-(1-carbamoylcyclopentyl)-6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidine
(3aS,6aS)-2-methanesulfonyl-5-(oxane-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-3-methylthiophene-2-carboxamide
4-[1-(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethyl]morpholine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(thiophen-2-yl)propan-1-one
2-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
ethyl 4-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}piperazine-1-carboxylate
methyl (2S,4R)-4-(dimethylamino)-1-[(2-phenylphenyl)methyl]pyrrolidine-2-carboxylate
3-(diphenylmethyl)-N-(3-ethoxypropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
3-benzyl-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-1,2-oxazole-5-carboxamide
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)-2-methoxyacetamide
1-{4-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
2-(3-methoxypropyl)-8-[(1-methyl-1H-indol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3R,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]pyridin-2-amine
1-cyclopentyl-3-{2-[4-(4-hydroxyphenyl)piperazin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
2-methyl-4-(3-{4-[2-(pyridin-4-yl)ethyl]piperazine-1-carbonyl}phenyl)butan-2-ol
2-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
(2S,4R)-1-(2-methoxyethyl)-N-methyl-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-amido)pyrrolidine-2-carboxamide
2-(4-methylpentyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]morpholine
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
2-methyl-4-[5-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)thiophen-2-yl]but-3-yn-2-ol
(1S,5R)-3-[(4-methyl-1,3-thiazol-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
6-{[2-(ethanesulfonyl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
5-(2,3-dihydro-1-benzofuran-7-carbonyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
7-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]-1H-indole
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-({8-[(3-hydroxy-4-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
(cyclopropylmethyl)({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
4-(2-hydroxypropyl)-8-thia-4,6-diazatricyclo[7.6.0.02,7]pentadeca-1(9),2(7),5-trien-3-one
2-cyclopentyl-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(4aR,7aS)-4-(5-methylthiophene-2-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3,5,7-trimethyl-2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-1H-indole
N'-(2,5-dimethylphenyl)-N-[1-(1H-indol-1-yl)propan-2-yl]propanediamide
methyl (2S,4R)-1-[(2-ethoxyphenyl)methyl]-4-[3-(3-fluorophenyl)benzamido]pyrrolidine-2-carboxylate
2-[(5-methylpyrazin-2-yl)methyl]-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
7-[3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3,6,7-trimethyl-1-benzofuran-2-carboxamide
2,3-difluoro-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]benzamide
5-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
1-(7-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-3-propylpiperidine-3-carboxylic acid
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-1-methylpiperidine-2-carboxamide
6,8-dimethyl-N-(1-methylpiperidin-3-yl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-3-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}benzamide
2-(4-fluorophenyl)-4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]morpholine