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N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,4,6-trimethylpyrimidin-2-amine
1-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
4-{[(2-ethoxy-3-methoxyphenyl)methyl](methyl)amino}pyrimidine-5-carboxylic acid
methyl 4-{[cyclohexyl(pyridin-2-ylmethyl)carbamoyl]amino}benzoate
1-[4-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)piperidin-1-yl]ethan-1-one
(2S)-2-amino-4-[1-(3-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]butanoic acid
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrazole-4-carboxamide
(3S)-4-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,3-dimethylpiperazin-2-one
N3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-N1,N1-dimethylpiperidine-1,3-dicarboxamide
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
(3S,9aR)-8-(2,5-dimethylbenzenesulfonyl)-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}propanamide
3-methoxy-N-(1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
3-[1-(2,5-dihydro-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-(1H-imidazol-1-yl)-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
4-[6-(3-fluoro-4-phenylphenyl)pyridine-3-carbonyl]morpholine
5-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-1-[(2-chlorophenyl)methyl]azepan-2-one
1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
1-[1-(2-methoxyacetyl)piperidine-3-carbonyl]-4-phenylpiperidine-4-carbonitrile
6-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-(2-methylquinoline-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
methyl (2S)-2-(3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-2-phenylacetate
2-{[4-(2-fluoro-4-hydroxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
6-(4-methoxyphenyl)-7-methyl-2-(piperidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-(1H-1,2,3-benzotriazol-5-yl)-4,4-difluoropiperidine-1-carboxamide
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-(4-acetylphenyl)urea
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S)-2-amino-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-(4-hydroxyphenyl)-N-methylpropanamide
2-[benzyl({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]ethan-1-ol
N-[(3R,4R)-1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
4-[(dimethylamino)methyl]-1-[(4-phenylphenyl)methyl]piperidin-4-ol
[(4-{2-[4-(3,4-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
2-(1H-pyrazol-1-yl)-N-[2-(pyridin-3-yl)ethyl]butanamide
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-[(4-chlorophenyl)methyl]-N-(2-hydroxy-2-phenylethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-{[(thiophen-2-ylmethyl)carbamoyl]methyl}pyrrolidine-3-carboxylic acid
9-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-[(4-fluorophenyl)methyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(4aR,8aS)-6-(2,5-dimethoxybenzoyl)-1-[(4-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
7,7-dimethyl-2-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N,N-dimethyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}acetamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(1H-pyrazol-1-yl)benzamide
7-fluoro-3-methyl-N-[2-(pyridin-4-yl)ethyl]-1-benzofuran-2-carboxamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-[(diethylamino)methyl]-N-(1-methylpiperidin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide