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(2S,4S)-1-(cyclohexylmethyl)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-[2-(3-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
methyl 4-[({2-[5-oxo-1-(2-phenylpropyl)pyrrolidin-2-yl]ethyl}amino)methyl]benzoate
7-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2,3-dimethyl-1H-indole
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]benzamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-cyclopentyl-N-{3-[4-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]phenyl}acetamide
(5R)-5-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-2-one
N-[2-(3-methoxyphenyl)ethyl]-6-(1-phenylcyclopropanecarbonyl)-6-azaspiro[2.5]octane-1-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]propanamide
N-[(2R,3R)-2-methoxy-1'-(3-methylbut-2-enoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
2-methoxy-N-[1-(pyrazin-2-yl)propan-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-cyclobutanecarbonyl-1'-(pyrrolidine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1H-1,2,3-triazol-4-yl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(2E)-N-({7-[(2S)-2-acetamido-4-methylpentanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
3-(2-fluorobenzoyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(pyrrolidin-3-yl)ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
4-(3,4-diethoxyphenyl)-2-(furan-3-yl)-1H-imidazole
8-methoxy-2-methyl-4-(quinolin-7-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-1,2,3-triazole
3-(6-methoxynaphthalene-2-carbonyl)-1-(3-methylthiophene-2-carbonyl)piperidine
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
[1-(2,5-dimethylpyrimidin-4-yl)-3-[(3-methoxyphenyl)methyl]piperidin-3-yl]methanol
N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(piperidin-1-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-ol
1-{1-[5-(2-methylphenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}propan-1-one
methyl 4-{2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}butanoate
2-(2,3-dimethylphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
(2R,6S)-2,6-dimethyl-4-[4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-yl]morpholine
N-({7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-ethyl-N-[(5-methylfuran-2-yl)methyl]acetamide
4-hydroxy-2-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)pyrimidine-5-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N,N-diethyl-1,3-oxazole-4-carboxamide
N-{2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl})amine
1-benzyl-8-[(2-methoxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{2-[2-(1-phenylethyl)-1H-imidazol-1-yl]ethyl}pyridine
3,3-dimethyl-1-(2-oxo-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)urea
2-(morpholin-4-yl)-2-(pyridin-3-yl)-1-(thiomorpholin-4-yl)ethan-1-one
2-[2-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
3-[(2-fluorophenyl)formamido]-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]propanamide
1-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
ethyl 1-[2-(cyclohex-1-en-1-yl)acetyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-methyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-3,4-dihydropyrimidin-4-one
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(3-methoxyphenyl)methyl]methylamine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
N-(1-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
N-{2-[3-(phenoxymethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide