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1,5-diamino-4-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-2,3-dihydro-1H-pyrrol-3-one
2-({3-cyano-3-[(2E)-2,3-dihydro-1,3-benzothiazol-2-ylidene]-2-oxopropyl}sulfanyl)acetic acid
ethyl 2-amino-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate
ethyl 2-amino-5-oxo-1-phenyl-4,5-dihydro-1H-pyrrole-3-carboxylate
1,8-diamino-6-methoxy-3-(piperidin-1-yl)-2,7-naphthyridine-4-carbonitrile
1,8-diamino-6-methoxy-3-(morpholin-4-yl)-2,7-naphthyridine-4-carbonitrile
1,8-diamino-6-ethoxy-3-(piperidin-1-yl)-2,7-naphthyridine-4-carbonitrile
1,8-diamino-6-ethoxy-3-(morpholin-4-yl)-2,7-naphthyridine-4-carbonitrile
2-amino-4-(cyanomethyl)-6-(piperidin-1-yl)pyridine-3,5-dicarbonitrile
2-amino-4-(cyanomethyl)-6-(morpholin-4-yl)pyridine-3,5-dicarbonitrile
2-amino-4-(1-cyano-2-phenylethyl)-6-(morpholin-4-yl)pyridine-3,5-dicarbonitrile
2-amino-4-(1-cyano-2-phenylethyl)-6-(piperidin-1-yl)pyridine-3,5-dicarbonitrile
2-amino-4-[(1Z)-1-cyano-2-(4-methoxyphenyl)eth-1-en-1-yl]-6-(piperidin-1-yl)pyridine-3,5-dicarbonitrile
2-amino-4-[(1Z)-1-cyano-2-(4-methoxyphenyl)eth-1-en-1-yl]-6-(morpholin-4-yl)pyridine-3,5-dicarbonitrile
1,8-diamino-3,6-diethoxy-2,7-naphthyridine-4-carbonitrile
1,8-diamino-3,6-dimethoxy-2,7-naphthyridine-4-carbonitrile
2-[(2Z)-4-oxo-3,4-dihydro-2H-1,3-benzothiazin-2-ylidene]acetonitrile
ethyl 2-[(2Z)-4-oxo-3,4-dihydro-2H-1,3-benzothiazin-2-ylidene]acetate
4-chloro-2-[(2Z)-2,3-dihydro-1H-1,3-benzodiazol-2-ylidene]-3-oxo-4-phenylbutanenitrile
4-chloro-2-[(2Z)-2,3-dihydro-1,3-benzothiazol-2-ylidene]-3-oxo-4-phenylbutanenitrile
5,6-diamino-3-methyl-2-oxo-8-(piperidin-1-yl)-1H,2H,3H-pyrrolo[2,3-c]2,7-naphthyridine-9-carbonitrile
5,6-diamino-8-(diethylamino)-3-methyl-2-oxo-1H,2H,3H-pyrrolo[2,3-c]2,7-naphthyridine-9-carbonitrile
5,6-diamino-3-methyl-8-(morpholin-4-yl)-2-oxo-1H,2H,3H-pyrrolo[2,3-c]2,7-naphthyridine-9-carbonitrile
methyl 4-amino-3-(1,3-benzothiazol-2-yl)-1-phenyl-1H-pyrazole-5-carboxylate
methyl 4-amino-3-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-1-phenyl-1H-pyrazole-5-carboxylate
methyl 6-amino-5-cyano-2-(2-methoxy-2-oxoethyl)-4-(4-methoxyphenyl)-4H-pyran-3-carboxylate
methyl 6-amino-5-cyano-4-(4-fluorophenyl)-2-(2-methoxy-2-oxoethyl)-4H-pyran-3-carboxylate
2-[(1-hydroxy-2-oxo-2-phenylethyl)sulfanyl]acetic acid
5,6-diamino-2-(chloromethyl)-8-(piperidin-1-yl)-1H,2H-furo[2,3-c]2,7-naphthyridine-9-carbonitrile
5,6-diamino-2-(chloromethyl)-8-(morpholin-4-yl)-1H,2H-furo[2,3-c]2,7-naphthyridine-9-carbonitrile
5,6-diamino-2-(chloromethyl)-8-(diethylamino)-1H,2H-furo[2,3-c]2,7-naphthyridine-9-carbonitrile
5,6-diamino-2-ethyl-8-(piperidin-1-yl)-1H,2H-furo[2,3-c]2,7-naphthyridine-9-carbonitrile
5,6-diamino-2-ethyl-8-(morpholin-4-yl)-1H,2H-furo[2,3-c]2,7-naphthyridine-9-carbonitrile
5,6-diamino-8-(diethylamino)-2-ethyl-1H,2H-furo[2,3-c]2,7-naphthyridine-9-carbonitrile
2-(phenylamino)thieno[2,3-d][1,3]thiazole-5-carboxylic acid
2-{5,7-dimethyl-2-sulfanyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetic acid
2-chloro-N-(3-methoxyphenyl)-3-oxo-3-phenylpropanamide
N-(2H-1,3-benzodioxol-5-yl)-2-chloro-3-oxo-3-phenylpropanamide
2-chloro-N-{1,7,7-trimethylbicyclo[2.2.1]heptan-2-yl}acetamide
methyl 2,3-dibromobutanoate
4-chloro-6-(chloromethyl)-2-(methylsulfanyl)pyrimidine
N-(4-carbamothioylphenyl)furan-2-carboxamide
4-(2-bromoethoxy)benzene-1-sulfonamide
2-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]acetonitrile
4-(pyrrolidin-1-ylmethyl)benzonitrile
2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1-(3,4,5-trimethoxyphenyl)ethan-1-one
2-[1-(difluoromethyl)-1H-1,3-benzodiazol-2-yl]-1-(3,4,5-trimethoxyphenyl)ethan-1-one
4-(6-nitro-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)butanoic acid
3-amino-4-chloro-N-[3-(morpholin-4-yl)propyl]benzene-1-sulfonamide
N-{[4-(propan-2-yl)phenyl]methyl}cyclopropanamine