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N-ethyl-2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
2-{[ethyl(oxan-2-ylmethyl)amino]methyl}benzoic acid
1-(5-methanesulfonamido-2-methylphenyl)-3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]urea
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-(oxolane-2-carbonyl)piperazine
1-{2-[1-(4-fluoro-2-methylbenzenesulfonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-5-phenyl-1H-pyrazole-3-carboxamide
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
3-(3,4-dimethoxybenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazole-3-carboxamide
(3S,4S)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(2-methoxyphenoxy)acetamide
3-(4-chlorobenzoyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
3-(2-methoxyquinolin-3-yl)-N-methylpyrazin-2-amine
1-[(2S)-2-(dipropylamino)propanoyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-{4-cyclopentyl-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-(2-ethoxyethyl)pyrrolidin-3-yl]-2-(thiophen-3-yl)acetamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyridin-2-amine
(1R,3S)-7-(furan-3-ylmethyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
5-[6-(2-methoxyphenyl)pyridazin-3-yl]pyridin-3-amine
2-(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-(3-chlorophenyl)-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[3-oxo-9-(9H-purin-6-yl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylate
4-{[1-(methylcarbamoyl)butyl]carbamoyl}benzoic acid
4-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-N-methylpyridin-2-amine
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[(3S,4S)-3-hydroxy-4-(4-methylpiperidin-1-yl)pyrrolidin-1-yl]propan-1-one
3-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4R)-1-(4-fluoro-2-methylbenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
4-phenyl-1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}-1,2,3,6-tetrahydropyridine
(3S,5S)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
4-(2,4-dimethoxybenzoyl)-1,4-diazabicyclo[3.2.2]nonane
3-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
8-(5-chloro-2-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-({1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
4-{1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-3-yl}benzoic acid
N-{2-[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-3-carboxamide
1-(5-methoxy-2-{5-methylthieno[2,3-d]pyrimidin-4-yl}phenyl)-1H-pyrazole
8-methoxy-N-{2-[(pyridin-3-yl)amino]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
ethyl 1-(1-acetylpiperidin-4-yl)-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
4-{4-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-6-[1-(6-methyl-1,3-benzothiazol-2-yl)piperidin-3-yl]pyrimidin-4-ol
1-(4-{[(2,1,3-benzoxadiazol-5-ylmethyl)amino]methyl}phenoxy)-3-[benzyl(methyl)amino]propan-2-ol
(2S,3R)-2-amino-3-hydroxy-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}butan-1-one
1'-(5-methoxyfuran-2-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[5-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-(3-methoxyphenoxy)-3-{[4-methyl-4-(methylsulfanyl)pentan-2-yl]amino}propan-2-ol