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N,N-dimethyl-5-(3-methyl-3-phenylpiperidin-1-yl)-1,2,4-thiadiazol-3-amine
4-{[3-ethoxy-4-(propan-2-yloxy)phenyl]methyl}-2-(trifluoromethyl)morpholine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1H-pyrrole-2-carboxamide
2-methyl-6-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)pyrimidin-4-ol
2-(2-fluorophenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
methyl 4-{3-[(3,4-difluorophenyl)amino]piperidine-1-carbonyl}benzoate
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({[2-(ethylsulfanyl)ethyl]carbamoyl}amino)-2-methylbenzamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]-N-[3-(oxolan-2-yl)propyl]benzamide
4-(4-methyl-1H-pyrrole-2-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-(4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperazin-1-yl)ethan-1-one
3-[2-(4-acetylphenyl)-1H-imidazol-1-yl]-4-fluorobenzoic acid
1-[(3-methylphenyl)methyl]-4-(quinolin-4-ylmethyl)piperazin-2-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
6-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-chloro-N-[2-(cyclohex-3-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
8-[(2S)-2-amino-2-cyclopropylacetyl]-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(pyridin-3-yl)pyrimidin-4-amine
1-[1-(3-cyano-6-methylpyridin-2-yl)piperidin-3-yl]-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
N-({5-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
methyl (2S)-2-{[7-acetyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-4-methylpentanoate
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[2-(methylsulfanyl)ethyl]piperidine-4-carboxamide
9-[2-(difluoromethoxy)benzoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-(5-{[(3S)-3-acetamidopyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
3-{[1-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1H-1,2,3-triazol-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
1,3-dimethyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3R,4R)-4-(azepan-1-yl)-1-(1-phenylpiperidin-4-yl)piperidin-3-ol
5-(2,5-dimethylphenoxymethyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[1-(4-chlorophenyl)cyclobutyl]-1-ethyl-1H-pyrazole-4-carboxamide
2-(3-methyl-1H-pyrazole-5-carbonyl)-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-(1-benzothiophen-2-ylmethyl)-1-cyclopentyl-N-methyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-[(2R,3R,6R)-5-[(2-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-methoxypyridine-3-carbonitrile
3-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,9aR)-8-(4-methylbenzenesulfonyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2S,4S)-N-ethyl-4-(4-ethylbenzamido)-1-[2-(methylsulfanyl)acetyl]pyrrolidine-2-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-(1H-pyrazol-1-yl)butanamide
{[3-(furan-2-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
2-(4-{[(1H-indol-4-ylmethyl)(methyl)amino]methyl}piperidin-1-yl)ethan-1-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-N'-(2,4-dimethylphenyl)ethanediamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-hydroxy-6-(trifluoromethyl)pyridine-3-carboxamide
3-{1-[(1-hexylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-1-ol
N-{1-azabicyclo[2.2.2]octan-3-yl}-5-phenyl-1,2-oxazole-4-carboxamide
2-[(1-methyl-1H-indol-2-yl)methyl]-2,8-diazaspiro[4.5]decane
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide