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N-methyl-6-[(3-methylthiophen-2-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
3-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]-1-[6-(2-methoxyphenoxy)pyridin-3-yl]urea
5-{[5-(2,5-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1-methylpyrrolidin-2-one
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-ethyl-7-methoxy-4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
{2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-2-oxoethyl}urea
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
1-{1-[(2,6-dimethylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-(1H-indol-5-yl)-5-oxopyrrolidine-3-carboxylic acid
5-[3-(2-ethoxyethoxy)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(1S,5R)-6-[(5-methylfuran-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1,3-thiazol-4-yl)ethan-1-one
6-(isoquinolin-5-yl)-2-(morpholin-4-yl)pyrimidin-4-amine
N-{1-[1-(3,3,5,5-tetramethylcyclohexyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
(1S,2S)-N2-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}-2,3-dihydro-1H-indene-1,2-diamine
1-(2-oxo-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)azepan-2-one
7-chloro-3-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}methyl)-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
3-{1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
[4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1,4-oxazepan-6-yl]methanol
(3aR,6aR)-2-(2-amino-6-methoxypyrimidin-4-yl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
3-(4-phenoxybenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
methyl (2S)-2-{[3-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]formamido}propanoate
4-(1-benzofuran-2-ylmethyl)-2-(morpholin-4-ylmethyl)-1,4-oxazepane
ethyl 2-[(2R,3R)-2-hydroxy-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]acetate
(3S,4S)-1-(1,3-benzothiazol-2-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[4-(1H-pyrazol-5-yl)benzoyl]piperidine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
1-(5-phenyl-1,3-oxazole-4-carbonyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
5-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-butyl-1-methyl-4-[3-(thiophen-2-yl)propanoyl]piperazin-2-one
(2S,4R)-N,N-diethyl-4-(2-hydroxy-5-methylbenzamido)-1-propanoylpyrrolidine-2-carboxamide
2-({1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
4-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-N-(pyridin-3-yl)benzamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
5-ethyl-1'-(1-methyl-1H-indole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-methoxy-1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-indole-2-carboxamide
4-methyl-6-[(3R)-3-methylpiperazin-1-yl]-5-(prop-2-en-1-yl)pyrimidin-2-amine
[1-(3-fluoro-2-methoxybenzoyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
1-ethyl-N-[(2-methoxyphenyl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N'-(3-ethylphenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]butanediamide
N-[2-(2-methylpropanesulfonyl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-butyl-4-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-cyclopentylacetamide
(1S,5R)-3-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[(4-ethylpiperazin-1-yl)methyl]-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-1,2-oxazole-3-carboxamide