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(3S,4R)-4-(3-methoxyphenyl)-1-[4-(prop-2-en-1-yl)benzoyl]pyrrolidine-3-carboxylic acid
N-{3-[({[3-(2-methylphenyl)phenyl]methyl}amino)methyl]-5-(piperidine-1-carbonyl)phenyl}methanesulfonamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(oxolan-3-yl)pyridin-2-amine
(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
2-(2-chloro-6-fluorophenyl)-1-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-N-(pyrazin-2-yl)benzamide
N-(2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}quinolin-5-yl)acetamide
3-[4-(4-fluorophenyl)-4-hydroxypiperidine-1-carbonyl]-5-methoxybenzoic acid
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(methylamino)acetamide
(4aS,7aR)-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)amine
1-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}azepane-2-carboxamide
N-[2-(oxan-2-yl)ethyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
9-[(3,4-dimethylphenyl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-{[6-(2-methoxyphenyl)pyridazin-3-yl]amino}-4-methylpentanamide
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-(2-methyl-1H-1,3-benzodiazol-6-yl)-4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-1-phenylcyclohexane-1-carboxamide
1-methyl-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-cyano-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
7-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
1-{3-[(5-ethylpyrimidin-2-yl)amino]propyl}pyrrolidin-2-one
1-({[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}methyl)cyclohexan-1-ol
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetamide
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-methanesulfonylpiperidin-4-amine
2-(2-oxopyrrolidin-1-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
N,1-diethyl-3-(2-methylpropyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
(2S)-2-hydroxy-4-[4-phenyl-5-(pyridin-2-yl)-1H-imidazol-1-yl]butanoic acid
3-cyclopropyl-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclopentan-1-ol
1-[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(morpholin-2-yl)ethan-1-one
2-{1-[(2,6-dimethylphenyl)methyl]pyrrolidin-3-yl}benzoic acid
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
(3R,4R)-3-cyclobutyl-4-methyl-1-[3-(morpholin-4-yl)benzoyl]pyrrolidin-3-ol
5-methyl-6-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]pyrazine
5-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]quinoxaline
N-ethyl-4-[2-(propan-2-ylsulfanyl)acetamido]piperidine-1-carboxamide
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
1-methyl-2-{1-[3-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
2-benzyl-4-[(2-ethylpyrimidin-5-yl)methyl]morpholine
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
1-(furan-3-ylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide