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N-cyclopropyl-6-ethyl-N-[(2-methoxyphenyl)methyl]-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-methoxyphenyl)-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
N-[(4-fluorophenyl)methyl]-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(pyrazin-2-yl)acetamide
4-methyl-N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-1,3-oxazole-5-carboxamide
N-[3-(dimethylamino)-1-phenylpropyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
(2S)-4-methyl-2-[(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)formamido]pentanamide
6-oxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
ethyl 2-(4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}morpholin-3-yl)acetate
4-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1,3-thiazole-5-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methoxyethan-1-one
5-{[(2S,5R)-5-(morpholin-4-ylmethyl)oxolan-2-yl]methyl}-2-(pyridin-3-yl)-1,3-benzoxazole
1-(3-phenylpropyl)-N-[2-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
6-methyl-N-(2-phenoxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1S,5R)-6-benzyl-3-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[benzyl(methyl)amino]-3-[4-({[(3-ethyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-(2-chlorophenoxy)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]ethan-1-one
methyl(2-methylpropyl)({5-[(3-methylquinoxalin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amine
3-(2-fluorophenyl)-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-5-carboxamide
1-ethyl-4-(4-{4-[4-(4-fluorophenoxy)piperidin-1-yl]piperidin-1-yl}benzoyl)piperazine
(1-{[4-(4-chlorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-2-yl)methanol
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[(4-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
7-fluoro-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]quinazolin-4-amine
N,N-diethyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
5-ethyl-1'-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3,4-dimethylphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-one
4-{1-[4-(2,6-dimethoxypyrimidin-4-yl)piperazin-1-yl]-2-methylpropan-2-yl}morpholine
4-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzoic acid
4-(1H-pyrrol-1-yl)-2-[2-(trifluoromethyl)morpholine-4-carbonyl]phenol
1-(azepan-1-yl)-2-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
1-({[2-(4-chloro-1H-pyrazol-1-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
1-[2-(3-propoxypiperidin-1-yl)pyrimidin-4-yl]piperidin-4-ol
1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
3-[1-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)azetidin-3-yl]pyridine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(2,5-dimethylthiophene-3-sulfonamido)acetic acid
3-ethyl-6-[4-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
1-[2-(2-chlorophenyl)ethyl]-N,N-diethyl-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
7-(4-fluorobenzenesulfonyl)-2-methyl-2,7-diazaspiro[4.5]decane
N-[3-(2-acetamidoacetamido)phenyl]-2-methoxybenzamide
4-{2-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
2-{[1-(morpholin-4-yl)hex-5-en-2-yl]oxy}quinoxaline
3-methyl-6-[5-(1-methylpiperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridazine
N-cyclopentyl-4-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,2,3-thiadiazole-5-carboxamide
N,N-diethyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
2-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,3-dimethylbutan-1-one
4-(1-ethylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
(3aS,6aS)-1-[2-(2-methoxy-4-methylphenoxy)ethyl]-octahydropyrrolo[2,3-c]pyrrole
6-{5-[5-(hydroxymethyl)furan-2-yl]-4-phenyl-1H-imidazol-1-yl}-2-methylheptan-2-ol
(2S)-2-acetamido-N-methyl-4-(methylsulfanyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide