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2-[4-(benzenesulfonyl)piperazin-1-yl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
2-(adamantan-1-yl)-N-(1-ethoxy-2-methylpropan-2-yl)acetamide
4-phenyl-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
1-{4-[7-(methylsulfanyl)-3-{[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}quinolin-2-yl]piperazin-1-yl}ethan-1-one
5-ethyl-6-methyl-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
6-ethoxy-4-methyl-2-{4-[(5-methylfuran-2-yl)methyl]-1,4-diazepan-1-yl}quinazoline
4-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)benzoic acid
2-[4-(2-methoxyphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
(3S,4R)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[5-(furan-2-ylmethyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
2-{3-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
4-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
1-(2-fluorophenyl)-2,2-dimethyl-N-[3-(3-oxopiperazin-1-yl)propyl]cyclopropane-1-carboxamide
3-(2,3-dihydro-1H-isoindol-2-yl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzamide
5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]-4-[1-(thiophene-3-carbonyl)piperidin-3-yl]pyrimidine
(1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-2-yl)methanol
1-ethyl-5-[2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-(4-chloro-2-methoxyphenoxymethyl)-N-methyl-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[(2-chloro-5-methoxy-4-propoxyphenyl)methyl]-N-cyclopropylpiperazine-2-carboxamide
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(2-propyl-1H-1,3-benzodiazol-1-yl)propanamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
3-{1-[(2,4-difluorophenyl)carbamoyl]piperidin-3-yl}benzoic acid
3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-phenylpropanamide
2-[(prop-2-en-1-yl)amino]-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
(5S,9aS,9bS)-5-(2,3-difluorophenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl](methyl){[4-(pyridin-2-ylmethoxy)phenyl]methyl}amine
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-methoxy-N-{1-[1-(3-methoxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-ethoxy-3-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}pyridine
4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
4-(7-fluoro-2-methylquinoline-4-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-[(5-oxo-1-phenylpyrrolidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(4-methylpent-3-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-butyl-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-(3-phenylprop-2-yn-1-yl)acetamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidine-5-carboxamide
7-(4-hydroxy-4-phenylpiperidine-1-carbonyl)-3-methyl-3,4-dihydroquinazolin-4-one
5-{2-[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazol-3-ol
4-chloro-1-methyl-3-{1-[1-(1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-1H-indazole
(4aS,7aR)-1-[(3,5-dichlorophenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-chloro-2-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]quinoline
1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-4-(pyridin-3-ylmethyl)piperazine
4-methyl-6-(4-phenylpiperidin-1-yl)pyrimidin-2-amine
2-[1-benzyl-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
dimethyl(2-{[(5-methylthiophen-2-yl)methyl](oxolan-3-ylmethyl)amino}ethyl)amine
3-methyl-8-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-ethyl-1-[(1-methylpiperidin-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
N-[3-(3-chlorophenyl)phenyl]-1-(3-hydroxy-2,2-dimethylpropyl)piperidine-4-carboxamide
(3S,4S)-4-(dimethylamino)-1-[(8-methoxyquinolin-2-yl)methyl]pyrrolidin-3-ol