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6-bromo-N-cyclohexylpyridin-2-amine
1-(4-bromo-1,3-thiazol-2-yl)-4-methylpiperidine
1-(4-chloropyrimidin-2-yl)pyrrolidin-3-ol
4-chloro-2-(1H-pyrazol-1-yl)pyrimidine
[6-(oxolan-3-yloxy)pyridin-2-yl]boronic acid
[6-(dimethylamino)pyridin-2-yl]boronic acid
6-bromo-N,N-diethylpyridin-2-amine
[6-(diethylamino)pyridin-2-yl]boronic acid
[6-(2-oxo-1,2-dihydropyridin-1-yl)pyridin-2-yl]boronic acid
2-bromo-6-(3-methyl-1H-pyrazol-1-yl)pyridine
[6-(3-methyl-1H-pyrazol-1-yl)pyridin-2-yl]boronic acid
2-bromo-6-(4-methyl-1H-pyrazol-1-yl)pyridine
[6-(4-methyl-1H-pyrazol-1-yl)pyridin-2-yl]boronic acid
[6-(1H-imidazol-1-yl)pyridin-2-yl]boronic acid
[6-(4-methylpiperazin-1-yl)pyridin-2-yl]boronic acid
1-(4-bromo-1,3-thiazol-2-yl)-3-methylpiperidine
1-(4-bromo-1,3-thiazol-2-yl)-2-methylpiperidine
4-bromo-N,N-dimethyl-1,3-thiazol-2-amine
4-bromo-N,N-diethyl-1,3-thiazol-2-amine
4-bromo-2-(1H-imidazol-1-yl)-1,3-thiazole
4-bromo-2-tert-butyl-1,3-thiazole
4-bromo-2-(4-methyl-1H-pyrazol-1-yl)-1,3-thiazole
4-bromo-2-(3-methyl-1H-pyrazol-1-yl)-1,3-thiazole
[2-(3-methyl-1H-pyrazol-1-yl)-1,3-thiazol-4-yl]boronic acid
[2-(4-methyl-1H-pyrazol-1-yl)-1,3-thiazol-4-yl]boronic acid
[2-(1H-imidazol-1-yl)-1,3-thiazol-4-yl]boronic acid
[2-(diethylamino)-1,3-thiazol-4-yl]boronic acid
[2-(dimethylamino)-1,3-thiazol-4-yl]boronic acid
(1,3-thiazol-4-yl)boronic acid
(2-methyl-1,3-thiazol-4-yl)boronic acid
[2-(3-methylpiperidin-1-yl)-1,3-thiazol-4-yl]boronic acid
[2-(2-methylpiperidin-1-yl)-1,3-thiazol-4-yl]boronic acid
[5-(2-oxo-1,2-dihydropyridin-1-yl)pyrazin-2-yl]boronic acid
2-bromo-5-(cyclopentyloxy)pyrazine
2-bromo-5-propoxypyrazine
(5-hydroxypyrazin-2-yl)boronic acid
2-bromo-5-(4-methylpiperidin-1-yl)pyrazine
[5-(4-methylpiperidin-1-yl)pyrazin-2-yl]boronic acid
2-bromo-5-(3-methylpiperidin-1-yl)pyrazine
[5-(3-methylpiperidin-1-yl)pyrazin-2-yl]boronic acid
2-bromo-5-(2-methylpiperidin-1-yl)pyrazine
[5-(2-methylpiperidin-1-yl)pyrazin-2-yl]boronic acid
2-bromo-5-(4-methylpiperazin-1-yl)pyrazine
[5-(4-methylpiperazin-1-yl)pyrazin-2-yl]boronic acid
2-bromo-5-(2-methyl-1H-imidazol-1-yl)pyrazine
[5-(2-methyl-1H-imidazol-1-yl)pyrazin-2-yl]boronic acid
2-bromo-5-(1H-imidazol-1-yl)pyrazine
[5-(1H-imidazol-1-yl)pyrazin-2-yl]boronic acid
2-bromo-5-(3-methyl-1H-pyrazol-1-yl)pyrazine
[5-(3-methyl-1H-pyrazol-1-yl)pyrazin-2-yl]boronic acid