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ethyl 4-({[7-chloro-2-oxo-1-(2-phenoxyethyl)-1,2-dihydroquinolin-3-yl]methyl}amino)piperidine-1-carboxylate
5-{[1-(ethylcarbamoyl)piperidin-4-yl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}quinoline-3-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(2,4-dioxoimidazolidin-1-yl)-N-methylbenzamide
1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-methyl-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)urea
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-6-[(1-methyl-1H-indol-3-yl)methyl]-3-(2-methylphenyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(2-phenylbenzoyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
(3aS,6aS)-2-methyl-5-[(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyridine-2-carbonitrile
2-{4-[2-(2,5-dimethylphenyl)acetyl]morpholin-3-yl}acetic acid
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[2-(4-methoxyphenyl)ethyl]urea
1-cyclohexyl-5-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
6-(2-fluorophenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
3-({2-[1-(oxane-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}acetamide
1-(5-acetyl-2-ethoxyphenyl)-3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]urea
4-(2-ethylpyrimidine-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
5-[(4aR,8aR)-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridine-1-carbonyl]-2,1,3-benzoxadiazol-1-ium-1-olate
3-(2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
2-methoxy-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenol
1'-(2-hydroxy-4-methylpentanoyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-[3-(4-methylpiperazine-1-carbonyl)phenyl]urea
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-(3-methylphenoxy)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
2-(3-{[ethyl(2,2,2-trifluoroethyl)carbamoyl]amino}phenyl)acetamide
2-[4-(2,5-dioxo-4-propylimidazolidin-4-yl)piperidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
4-methyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pentanamide
5-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-6-methoxy-3-methyl-N-(propan-2-yl)-1-benzofuran-2-carboxamide
7-(cyclopropylmethyl)-2-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-{[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzonitrile
N-{[7-fluoro-5-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenoxyacetamide
1-[(5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}furan-2-yl)methyl]-4-methylpiperidine
N-ethyl-3-{2-[methyl(pyridin-4-ylmethyl)amino]acetamido}-N-phenylbenzamide
4-{3-[1-(4-chlorophenyl)cyclopentyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-imidazole
N-(1-phenylpiperidin-4-yl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-cyclohexyl-1-[2-(morpholin-4-yl)ethyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
3-[2-(2,6-difluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
2-cyclopentyl-9-(2,4-dimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[5-methoxy-2-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[4-(propan-2-yl)phenyl]methyl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2-fluoro-5-methylphenoxy)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylic acid
N-[3-(3-methylphenyl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-3-carboxamide
3-cyclopropyl-5-(3-methylphenoxymethyl)-1H-1,2,4-triazole
1-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
N-(2-chloro-5-sulfamoylphenyl)-3-propoxypiperidine-1-carboxamide
1-[2-(2-chlorophenyl)ethyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
[(4-ethoxyphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine