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2-cyclohexyl-5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)pyrimidine
2-(3-methylpyrazin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
(4aS,7aR)-1-(3-chloro-4-fluorobenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-(morpholin-3-yl)ethan-1-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)pyridine-2-carboxamide
1-(3-methoxyphenyl)-4-(3-methoxypyrazin-2-yl)piperazin-2-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-oxobutanamide
N-[(2S,4R,6S)-2-ethyl-6-(2-fluoro-4-methoxyphenyl)oxan-4-yl]acetamide
3-[1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)piperidin-2-yl]pyridine
2-[4-phenyl-5-(propan-2-yl)-1H-imidazol-1-yl]-1-(piperazin-1-yl)ethan-1-one
N-[(6-methylquinolin-5-yl)methyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-N'-(4-methylphenyl)propanediamide
[(3S,5R)-1-(4-chloro-2-fluorobenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
methyl 2-({[2-(difluoromethoxy)phenyl]methyl}amino)pyridine-4-carboxylate
6-methyl-2-({[1-(pyrazin-2-yl)piperidin-3-yl]amino}methyl)quinolin-4-ol
2-(5-{[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl)pyridine
N-[(5-methylpyrazin-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(4aS,8aR)-1-(2-aminoethyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carboxamide
N-[3-(2-oxoimidazolidin-1-yl)phenyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidine
2-[4-(3-fluoropyridin-2-yl)-1H-pyrazol-1-yl]-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
1-(oxan-4-yl)-4-[4-(piperidin-1-ylmethyl)benzoyl]piperazine
4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
{1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]ethyl}dimethylamine
2-(4-fluorophenyl)-2-hydroxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{2-[1-(2,6-difluoro-4-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
1-[(3-fluorophenyl)methyl]-4-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)piperazin-2-one
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-(1,2-oxazol-5-ylmethyl)-2-phenylacetamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}propanamide
N-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-N-methyloxan-4-amine
2-methyl-4-(2-methylphenyl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(oxane-2-carbonyl)piperidine
ethyl 4-(5,6,7,8-tetrahydroquinoline-3-amido)piperidine-1-carboxylate
1-{4-[(dimethylamino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
2-(6-cyclopropylpyrimidin-4-yl)-N,N-bis(propan-2-yl)benzamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[2-(3-fluorophenyl)ethyl]piperidine
{4-[3-(azepan-1-ylmethyl)benzoyl]-1,4-oxazepan-6-yl}methanol
4-(4-ethoxy-3-methylphenyl)-N-[1-(furan-2-yl)ethyl]butanamide
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-3-(3-methylphenyl)-1H-pyrazole
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
5-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-4,6-dimethylpyrimidin-2-amine
3-hydroxy-3-{[(3-hydroxy-2,2-dimethylpropyl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
5-(7-fluoro-3-methyl-1-benzofuran-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
2-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
2-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(1R,5R)-N-benzyl-3-(dimethylsulfamoyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-cyclopentyl-3-(2-methoxyphenyl)-3-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]pyrrolidine-2,5-dione
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one