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1-(2-cyclohexylethyl)-3-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N-(1,2,3,4-tetrahydronaphthalen-2-yl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-(1-benzyl-4-hydroxypiperidin-4-yl)-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
N-methyl-4-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidine-1-carbonyl]pyridin-2-amine
N-[(3-ethoxyphenyl)methyl]-N-ethyl-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
11-[(1,3-benzothiazol-2-ylmethyl)amino]-4-[(2-fluorophenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[1-(3-phenylphenyl)piperidin-4-yl]-4-(prop-2-en-1-yl)piperazine
N-cyclopropyl-2-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]acetamide
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
2,3,5,6-tetramethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)benzamide
4-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}pyrimidine
3-(4-hydroxyphenyl)-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
N-(1-{[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)acetamide
2-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]methyl}-4-hydroxyquinoline-6-carboxamide
N-methyl-2-{3-oxo-2-azaspiro[4.5]decan-2-yl}-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
5-methyl-N-{4-[2-(1H-1,2,4-triazol-1-yl)acetamido]phenyl}furan-2-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(3,5-dimethyl-1H-pyrazol-1-yl)butanamide
2-[(4-methoxyphenyl)methyl]-6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-methyl-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-cyclohexylurea
2-{[4-(4-methoxyphenyl)-5-(4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-(2,5-dioxoimidazolidin-1-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
6-[(2,3-dihydro-1H-inden-1-yl)amino]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
7-(3-chloro-5-fluorobenzoyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N3-cycloheptyl-1-cyclopropyl-4-oxo-N5-[(4-phenyloxan-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(5-acetylthiophen-3-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
N-[(1-methylpyrrolidin-3-yl)methyl]-N'-[2-(methylsulfanyl)phenyl]butanediamide
1-(4-acetylpiperazin-1-yl)-3-(4-chlorophenyl)-3-phenylpropan-1-one
2-cyclopentyl-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-ethoxy-5-(2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrimidin-4-yl)benzoic acid
3-hydroxy-3-{[methyl(oxan-4-yl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-(pyrrolidin-3-yl)acetamide
N-[(5-chloro-2-ethoxyphenyl)methyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-methylpropanamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
N-(2,3-dihydro-1H-inden-2-yl)-3-[(2-methylpropyl)amino]-5-[(propan-2-yl)sulfamoyl]benzamide
1-acetyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
[(4-methoxy-3-methylphenyl)methyl]({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amine
1-{1'-[2-(propylsulfanyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methoxypyrimidine
(3aS,6aS)-2-[(4-chlorophenyl)methyl]-5-cyclopentanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidine
9-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(furan-3-ylmethyl)-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
9-methoxy-4-[(8-methoxyquinolin-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine
1-{[2-({[6-(morpholin-4-yl)pyrimidin-4-yl]amino}methyl)phenyl]methyl}pyrrolidin-2-one
5-{2-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}imidazolidine-2,4-dione
({5-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine