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methyl (2S,4S)-1-[(2,4-dimethylphenyl)methyl]-4-(pyridine-2-amido)pyrrolidine-2-carboxylate
N-[1-(6-ethyl-2-methylquinoline-4-carbonyl)piperidin-4-yl]pyrimidin-2-amine
4-methyl-2-oxo-5-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile
2-amino-6-(2,2-dimethyloxan-4-yl)-4-(2-methoxypyrimidin-5-yl)-5-methylpyridine-3-carbonitrile
N-(2,4-dimethoxyphenyl)-3-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]propanamide
2-{5-[1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
2-(3-chloro-4-fluorobenzoyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
5-(2H-1,3-benzodioxol-5-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,2,4-triazin-3-amine
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-[6-(dimethylamino)pyridine-3-carbonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(1-hydroxy-2-methylpropan-2-yl)-5-methyl-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-(2-methoxyethyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-methyl-1-{2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(naphthalen-2-ylmethyl)-1,4-diazepan-5-one
1-methyl-4-phenyl-N-(quinolin-3-ylmethyl)piperidine-4-carboxamide
3-chloro-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
(3aR,6aR)-2-cyclopentanecarbonyl-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[1-(5-chloro-2-methoxybenzenesulfonyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-(5-{[(cyclopropylmethyl)sulfanyl]methyl}-1,2,4-oxadiazol-3-yl)-6-methylpyridazine
2-(butylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-acetyl-N-[(3-fluoro-4-methoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
6-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-9H-purine
3-[({[1-(4-fluorophenyl)cyclopentyl]methyl}amino)methyl]piperidin-3-ol
3-[2-(dimethylamino)ethyl]-8-[2-(2-methoxyphenyl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-2-(1H-indol-1-yl)ethan-1-one
(5R)-5-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrrolidin-2-one
2-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methylphenol
N-methyl-5-[(methylsulfanyl)methyl]-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}furan-2-carboxamide
N-benzyl-N,1-dimethyl-5-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(5-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}furan-2-yl)methanol
3-cyclohexyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-1H-pyrazole-4-carboxamide
8-{[4-(2-ethylpiperidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
[1-(3,5,7-trimethyl-1H-indole-2-carbonyl)azepan-2-yl]methanol
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-{4-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
(2S,4S)-N-ethyl-1-(furan-2-ylmethyl)-4-[2-(2-methylphenyl)acetamido]pyrrolidine-2-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
dimethyl[2-({[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(2-methylphenyl)methyl]amino)ethyl]amine
1-ethyl-8-[(3-hydroxyphenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[(3,5-dimethoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-[(2-methylphenyl)sulfanyl]-1-(oxolane-2-carbonyl)piperidine
[1-(1H-imidazol-1-yl)propan-2-yl]({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amine
2-[1-(2-methylpropyl)-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
3-(2,3-dihydroxypropyl)-3-methyl-1-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
2-{[(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-(4-fluorophenyl)-3-phenylpropanamide
5-{[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-benzyl-N-methyl-3-[1-(thiophene-2-sulfonyl)piperidin-4-yl]propanamide
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
ethyl 3-[(3-chlorophenyl)methyl]-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylate