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2-{4-methyl-6-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]pyrimidin-2-yl}phenol
2-cyclopentyl-N-[1-methyl-2-(oxolan-2-yl)-7-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-5-yl]acetamide
2-(2-methyl-5-phenylfuran-3-yl)-6-(piperidin-3-yl)-3,4-dihydropyrimidin-4-one
[(3-chloro-4,5-diethoxyphenyl)methyl]({2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})methylamine
2-[(3,4-dimethoxyphenyl)methyl]-6-[2-(methoxymethyl)piperidine-1-carbonyl]-1,3-benzoxazole
3-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinoxalin-2-one
5-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxylic acid
2-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-{4-chloro-2-[(3-hydroxyazetidin-1-yl)methyl]-6-methoxyphenoxy}propanoic acid
N-[2-(azepan-1-yl)-2-phenylethyl]-4-chloro-1-methyl-1H-pyrazole-3-carboxamide
1-(pyrazin-2-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
methyl (2S,4S,5R)-5-(2-chlorophenyl)-4-[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylate
N-cyclopropyl-2-({1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
4-benzoyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,4R)-4-(3-fluorophenyl)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
8-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-(trifluoromethyl)benzamide
3-chloro-5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-tert-butyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
4-(4-fluorophenoxy)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
1-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)isoquinoline
2-[5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]acetic acid
{5-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-propoxypropan-1-one
1-cyclohexyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)piperidine-3-carboxamide
5-(2-methylfuran-3-carbonyl)-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3aS,6aS)-2-[(3-fluoro-2-methylphenyl)methyl]-5-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-butyl-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
(2S)-2-amino-3-(4-hydroxyphenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
4-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridin-1-ium-1-olate
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
2-(2-{[(2-propyl-1,3-thiazol-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-(2-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
N-[(3-chlorophenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-6-(oxan-4-yl)-3,4-dihydropyrimidin-4-one
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
4-(cyclopropylmethyl)-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid
(1R,9aR)-1-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
2-ethyl-N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-4-methyl-1,3-thiazole-5-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N1,N1-dimethyl-N3-[2-(2-methyl-1H-indol-3-yl)ethyl]piperidine-1,3-dicarboxamide
N-({1-[2-(4-fluorophenoxy)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
1-amino-N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}cyclopropane-1-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-(oxan-2-ylmethyl)acetamide
3-({3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}propanamide