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5-(3-methoxyphenyl)-N-[2-(pyridin-3-yloxy)propyl]-1,2,4-triazin-3-amine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
6-(4-chlorophenyl)-N,N-bis(2-hydroxyethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(1-{1-[(2,3,4-trifluorophenyl)methyl]piperidin-4-yl}ethyl)morpholine
N-methyl-1-(propan-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}piperidine-4-carboxamide
N-[3-(furan-2-yl)phenyl]-2-oxo-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
4-(4-fluorophenyl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
3-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[4-(3-fluorophenyl)oxan-4-yl]methyl})amine
2-ethyl-9-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-ethyl-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pentan-1-one
4-[(2-chloro-6-fluorophenyl)methyl]-6-(cyclopropylmethoxy)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-methyl-5-(propan-2-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)ethyl]acetamide
N-[2-(2,3-dimethoxyphenyl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-[(3-methylthiophen-2-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yloxy)-4-methoxyphenyl]methyl}pyrrolidine
N4-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-6-methylpyrimidine-2,4-diamine
(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
N-methyl-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(propan-2-yl)acetamide
4-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-2-methoxypyridine-3-carbonitrile
2-{5-[1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(4-fluorophenoxy)ethan-1-one
methyl 6-(3-fluorobenzoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl 4-{1-[(6-ethoxyquinolin-2-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-(morpholin-3-yl)ethan-1-one
8-(4-methylpyridine-3-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
7-(2-methylphenyl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(difluoromethoxy)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-3-chloro-1,2-dihydropyridin-2-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
4-(cyclopropylmethyl)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1,4-diazepan-5-one
7-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
2-{3-cyclopropyl-5-[2-(pyrazin-2-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
5-methoxy-2-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-4H-pyran-4-one
6-(ethylamino)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
1-methyl-3-({4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-indole
2,2-dimethylpropyl N-[(3R,5S)-5-[(3-hydroxyadamantan-1-yl)carbamoyl]pyrrolidin-3-yl]carbamate
methyl 3-[3-(3-hydroxypiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
2-[3,5-dimethyl-1-(pyridin-4-yl)-1H-pyrazol-4-yl]phenol
3-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)-N-(1,3-thiazol-2-yl)propanamide
4-ethyl-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1,2,3-thiadiazole-5-carboxamide
7-methyl-4-(3-methylphenyl)-6-(3-methylpyridine-2-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
(3aS,7aR)-5-methyl-2-(4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid