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2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
1,3-dimethyl-6-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
2-(4-{[8-methoxy-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenoxy)ethan-1-ol
(2S,4R)-4-amino-1-(5-ethoxy-2-methyl-1-benzofuran-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(3-hydroxyadamantan-1-yl)-3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamide
N-[(4-methyloxan-4-yl)methyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2S)-1-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidine-2-carboxamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
N-(2,5-dimethylphenyl)-3-[(1-methoxypropan-2-yl)amino]propanamide
methyl 3-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propanoate
1-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-amino-4-(1,2-dimethyl-1H-imidazol-5-yl)-6-(1-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-(2-methylphenyl)-5-{1-[1-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}pyrimidine
N4,N4,5-trimethyl-N2-[2-(4-methylpiperazin-1-yl)butyl]pyrimidine-2,4-diamine
(4aS,7aR)-1-(cyclopropanesulfonyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1-(propan-2-yl)piperidine
3-[2-(morpholin-4-ylmethyl)phenyl]-1-(1,2,3,4-tetrahydronaphthalen-1-yl)urea
methyl 9-(cyclopentyloxy)-3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-N-methyl-2-oxo-N-phenylacetamide
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(dicyclopropylmethyl)methylamine
1-[1'-(6-methyl-2-propylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
5-methyl-N-[(1r,4r)-4-hydroxycyclohexyl]-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3,3-dimethyl-1-(2-methyl-6-propylpyrimidin-4-yl)-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-1,4-dithiepan-6-amine
2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(oxane-4-carbonyl)-3-phenylpiperazine
1-cyclopropanecarbonyl-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-4-carboxamide
8-[3-(methylsulfanyl)propanoyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{4-[(3,5-dimethyl-1H-indol-2-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
5-(3,4-difluorophenoxymethyl)-N-ethyl-N-(2-methoxyethyl)-1,2-oxazole-3-carboxamide
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3-{[(6-methylpyridin-2-yl)methyl]amino}phenyl)pyrrolidin-2-one
N-[(1R,3R)-3-aminocyclopentyl]-1-benzyl-4-phenylpiperidine-4-carboxamide
3-[(4aR,7aS)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(3S,4R)-1-(1,4-dithiepan-6-yl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(4aR,7aS)-1-methyl-4-[3-(1H-pyrazol-1-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4-propylpyrrolidine-3-carboxylic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(propane-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[2-(2-methyl-1,4-oxazepane-4-carbonyl)pyridin-4-yl]methanol
5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2,1,3-benzoxadiazole
9-(4-methylpyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-N-(2-phenylethyl)piperidine-1-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[4-(hydroxymethyl)oxan-4-yl]benzamide
2-[5-(4-ethylpiperazin-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-indole-6-carboxamide
5-{3-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
2-(4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}morpholin-3-yl)-N-methylacetamide
(3S)-3-ethyl-4-[4-(3-fluorophenyl)benzoyl]morpholine
5-cyclopropanecarbonyl-1'-(pyridin-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]