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2-[(2R,5S)-5-(methanesulfonamidomethyl)pyrrolidin-2-yl]-N-methylacetamide
1-{2-[2-(6-chloropyrazin-2-yl)ethyl]piperidin-1-yl}ethan-1-one
1-{2-[2-(5-bromopyrazin-2-yl)ethyl]piperidin-1-yl}ethan-1-one
1-{4-[(6-chloropyridazin-3-yl)methyl]piperidin-1-yl}ethan-1-one
1-{4-[(6-chloropyridazin-3-yl)methyl]azepan-1-yl}ethan-1-one
1-[4-(6-chloro-2-methylpyrimidin-4-yl)piperidin-1-yl]-2,2-dimethylpropan-1-one
1-{4-[(6-chloropyrazin-2-yl)methyl]piperidin-1-yl}ethan-1-one
1-{4-[(3-chloropyrazin-2-yl)methyl]piperidin-1-yl}ethan-1-one
1-{4-[(3-chloropyrazin-2-yl)methyl]azepan-1-yl}ethan-1-one
1-[3-(6-chloropyrazin-2-yl)piperidin-1-yl]ethan-1-one
2-(3-chloropyrazin-2-yl)-N,N-dimethylpyrrolidine-1-sulfonamide
1-[3-(6-chloro-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-methoxyethan-1-one
3-(3-chloropyrazin-2-yl)-N,N-dimethylpiperidine-1-sulfonamide
1-{4-[(6-chloropyrazin-2-yl)methyl]azepan-1-yl}ethan-1-one
1-{2-[2-(6-chloropyrimidin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
1-[4-(6-chloropyrazin-2-yl)piperidin-1-yl]ethan-1-one
4-[(2-chloropyridin-4-yl)methyl]-1-methanesulfonylazepane
2-chloro-4-[2-(1-methanesulfonylpyrrolidin-2-yl)ethyl]pyridine
2-chloro-4-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]pyridine
4-[(3-chloropyrazin-2-yl)methyl]-1-methanesulfonylazepane
4-[(6-chloropyrazin-2-yl)methyl]-1-methanesulfonylazepane
1-[2-(5-bromo-4-methyl-1,3-thiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
1-[3-(5-bromo-4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
1-[3-(3-chloropyrazin-2-yl)piperidin-1-yl]ethan-1-one
2-bromo-6-[1-(propan-2-yl)pyrrolidin-2-yl]pyridine
2-bromo-6-[1-(propan-2-yl)piperidin-3-yl]pyridine
2-bromo-6-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}pyridine
4-[(6-bromopyridin-2-yl)methyl]-1-(propan-2-yl)azepane
2-chloro-4-[1-(propan-2-yl)piperidin-4-yl]pyridine
2-chloro-4-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}pyridine
4-[(3-chloropyrazin-2-yl)methyl]-1-(propan-2-yl)azepane
4-[(5-bromopyrazin-2-yl)methyl]-1-(propan-2-yl)azepane
4-[(6-chloropyridazin-3-yl)methyl]-1-(propan-2-yl)azepane
4-chloro-6-methyl-2-[1-(propan-2-yl)piperidin-4-yl]pyrimidine
4-chloro-2-methyl-6-[1-(propan-2-yl)piperidin-3-yl]pyrimidine
4-[(2-chloropyridin-4-yl)methyl]-1-(propan-2-yl)azepane
tert-butyl 4-(5-bromo-4-methyl-1,3-thiazol-2-yl)piperidine-1-carboxylate
4-[(6-bromopyridin-2-yl)methyl]-1-methylazepane
4-[(2-chloropyridin-4-yl)methyl]-1-methylazepane
2-chloro-6-(1-methylpiperidin-4-yl)pyrazine
4-chloro-2-methyl-6-(1-methylpiperidin-4-yl)pyrimidine
4-chloro-6-{2-[1-(propan-2-yl)pyrrolidin-2-yl]ethyl}pyrimidine
2-chloro-4-[2-(1-methylpiperidin-2-yl)ethyl]pyridine
4-chloro-2-methyl-6-[1-(propan-2-yl)piperidin-4-yl]pyrimidine
3-[(6-chloropyridin-3-yl)methyl]-N,N-dimethylpyrrolidine-1-sulfonamide
3-[(6-bromopyridin-2-yl)methyl]-N,N-dimethylpyrrolidine-1-sulfonamide
1-{3-[(2-chloropyridin-4-yl)methyl]piperidin-1-yl}ethan-1-one
1-{4-[(2-chloropyridin-4-yl)methyl]piperidin-1-yl}ethan-1-one
1-{3-[(6-bromopyridin-2-yl)methyl]pyrrolidin-1-yl}-2,2-dimethylpropan-1-one
1-{4-[(6-chloropyridin-3-yl)methyl]azepan-1-yl}ethan-1-one