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2-[methyl(pyridin-3-ylmethyl)amino]-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]ethan-1-one
(1S,6R)-3-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3,9-diazabicyclo[4.2.1]nonane
2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpiperazine-1-carboxamide
5-(4-fluoro-2-methylbenzoyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
9-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1R,3S)-7-(2,3-dimethyl-1H-indole-7-carbonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
5-{1-[2-(3,5-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-(3-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-methoxy-3,4-dihydroquinazolin-4-one
5-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-3,4-dihydropyrimidin-4-one
1-(2H-1,3-benzodioxole-5-carbonyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
1-{3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(1H-pyrazol-1-yl)propan-1-one
(4aR,7aS)-1-benzyl-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-4-cyclopropyl-1-(dimethylcarbamoyl)pyrrolidin-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
1-{2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N6-cyclopentyl-N5-methyl-N5-[4-(morpholin-4-yl)butyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
[(3R,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(pyridine-2-carbonyl)piperidin-3-yl]methanol
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-hydroxy-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
3-(4-methoxyphenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
6-(3-fluoro-4-methoxyphenyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}imidazo[2,1-b][1,3]thiazole
(1R,5R)-3-(dimethylsulfamoyl)-N-(3-methylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-benzyl-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
{4-[(4-chlorophenyl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}methanol
(3S,9aR)-3-[(benzyloxy)methyl]-8-(4-fluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
ethyl 3-(3-phenylpropyl)-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-3-carboxylate
[(3R,4S)-1-(9H-fluoren-2-ylmethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine-1-carboxamide
N1-{5-[2-(dimethylamino)ethyl]-1,3,4-thiadiazol-2-yl}-N4-(furan-2-ylmethyl)piperidine-1,4-dicarboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,6-difluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
(1R,5S,8S)-3-{1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}-3-azabicyclo[3.2.1]octan-8-ol
2-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
1-(2-methoxy-5-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
8-(1,3-dihydroxypropan-2-yl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-methyl-1H-pyrazol-5-yl)-2-[4-(9H-purin-6-yl)-1H-pyrazol-1-yl]acetamide
1-cyclobutanecarbonyl-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
7-(2-methoxypyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
ethyl 2-{1-[5-(4-acetylphenoxymethyl)-1,2-oxazol-3-yl]-N-methylformamido}acetate
2-(2-hydroxyphenoxy)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(4-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}phenyl)acetic acid
1-{5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
3,5-dimethyl-1-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azetidin-3-yl)-1H-pyrazole
N-phenyl-3-[1-(thiolan-3-yl)piperidin-4-yl]propanamide
3-{[(5-fluoro-3-methyl-1H-indol-2-yl)methyl](methyl)amino}-N-methylbutanamide
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(quinoxalin-5-ylmethyl)piperidin-3-yl]propan-1-one
N-[2-(1,3-benzoxazol-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1'-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one