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(4aS,7aR)-4-[(4-hydroxy-3-methylphenyl)methyl]-6,6-dioxo-N-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-methyl-N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-1,3-thiazole-4-carboxamide
2-{[4-(1H-imidazol-1-yl)phenyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(4-fluorophenyl)-4-{1-[(4-methylphenyl)methyl]piperidin-3-yl}piperazine
8-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-1-methyl-3-propyl-1H-pyrazole
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-hydroxypyrazine-2-carboxamide
(3S,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(methylsulfanyl)-N-(propan-2-yl)pyridine-3-carboxamide
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
(2-{[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
2-{5-[2-(methylamino)pyridine-4-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
{4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-1,4-oxazepan-6-yl}methanol
3-{1-[1-(1-methyl-1H-imidazol-2-yl)butyl]-4-phenyl-1H-imidazol-5-yl}pyridine
4-cyclobutyl-N,6-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidin-2-amine
2-chloro-4-[3-(propanamidomethyl)phenyl]benzamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(9H-purin-6-yl)piperazin-2-yl}ethan-1-ol
N-[1-(methylcarbamoyl)cyclohexyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}methyl)phenoxy]propan-2-ol
(1R,6S)-N-butyl-6-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}cyclohex-3-ene-1-carboxamide
2-(2-methoxypyrimidine-5-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}but-3-en-1-one
4-methyl-2-(methylamino)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,3-thiazole-5-carboxamide
methyl (2S)-2-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)-2-phenylacetate
2-(3-methoxyphenyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
1-{[4-(methylsulfanyl)phenyl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
5-butyl-1'-(5-ethyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 1-{9-methoxy-3-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
(3aS,6aS)-5-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(3-methoxyphenyl)-5-methyl-4-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
(2R,3R,6R)-5-(1,3-benzothiazole-6-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[1-(2-hydroxybutyl)-5-[(2-oxopyrrolidin-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
N-[4-(2-fluorophenoxy)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
(2R,3R)-3-({[3-(dimethylamino)phenyl]methyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-methoxy-1-{4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
2-{4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
N-{4-[2-(6-chloropyridin-3-yl)acetamido]-2-methylphenyl}-2,2-dimethylpropanamide
4-[(2S,4R)-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidine-2-carbonyl]morpholine
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyrrolidin-1-yl)benzamide
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-(morpholin-4-yl)cyclohexane-1-carboxamide
(2S)-4-{[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}-2-hydroxybutanoic acid
N-({1-[(2E)-2-methylpent-2-en-1-yl]piperidin-4-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
(4aS,7aR)-1-[(2-methoxyphenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,5R,6S,7aS)-2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-octahydro-1H-isoindole-5,6-diol
N-methyl-N-{[5-(4-phenyl-1H-imidazol-5-yl)furan-2-yl]methyl}methanesulfonamide
N-[(1S)-1-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl]acetamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-3,5-dimethyl-1H-pyrrole-2-carboxamide
4-(5-{[3-(pyridin-2-yl)propyl]carbamoyl}pyridin-2-yl)morpholine-2-carboxamide