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1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(1-methylcyclopropyl)propan-1-one
(2S)-2-phenyl-2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}acetamide
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
3-[(dimethylamino)methyl]-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]ethan-1-one
methyl 3-[4-(methoxycarbonyl)benzoyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2,6-dimethoxypyridin-3-yl)-2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carboxamide
1-tert-butyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
N,N,4-trimethyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyrimidin-2-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[methyl(propyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
9-[5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]-6-oxa-9-azaspiro[4.5]decane
3-[1-(3,5-dichloro-4-methylbenzoyl)piperidin-4-yl]-1,3-oxazolidin-2-one
N-[(3R,4S)-1-cyclopentyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
5,6-dimethyl-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,1,2,5-tetramethyl-1H-pyrrole-3-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
1'-(5-ethyl-1,3,4-thiadiazol-2-yl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]-2-{3-[4-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}acetamide
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyrrolidine-1-carbonyl)piperidine
4-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
1-(2-methyl-1,3-thiazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-[2-(4-sulfamoylphenyl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
(2S,4R)-N-ethyl-4-{[(4-fluorophenyl)methyl]amino}-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
3-[5-(3-phenoxypropyl)-1H-1,2,4-triazol-3-yl]pyridine
N-methyl-5-oxo-1-phenyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,5-dihydro-1H-pyrazole-3-carboxamide
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
3-methyl-8-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl (2S,4R)-1-[(2,5-dimethoxyphenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
1-[(4-methoxyphenyl)methyl]-3-(3-methoxypropyl)-3-(1-methylpiperidin-4-yl)urea
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-(5-methyl-1,3-benzoxazol-2-yl)piperidin-4-amine
N-[(2,4-dichlorophenyl)methyl]-2,8-diazaspiro[4.5]decane-2-carboxamide
2-{2-[(2-phenylazetidin-1-yl)methyl]phenoxy}ethan-1-ol
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-[3,3-dimethyl-1-(pyrrolidin-1-yl)butan-2-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
1-[2-methoxy-4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-(2,6-dimethoxypyridine-3-carbonyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-cyclopentylacetamide
2-(dimethylamino)-7-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{3-[5-(5-ethyl-1,2-oxazole-3-carbonyl)-3-(piperidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]propyl}pyridine
(1S,5R)-6-[4-(propan-2-yloxy)benzoyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-methyl-1,3-thiazol-4-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethan-1-one
1-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperidine-3-carbonitrile
(1R,3S)-3-amino-N-[(2,3-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)cyclohexane-1-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(1H-imidazol-2-yl)benzamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
5-methyl-4-[1-(oxan-4-yl)piperidin-3-yl]-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidine
1-(4-chlorophenyl)-3-(propan-2-yl)-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazole
1-(1-butanoylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-2-[4-(oxolan-2-ylmethyl)piperazin-1-yl]pyrimidine
N-[1-(furan-2-yl)ethyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine