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N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-5-methyl-1,3-oxazole-4-carboxamide
methyl 2-{[(2,3-difluoro-6-methoxyphenyl)methyl]amino}pyridine-4-carboxylate
2-(2-methoxyphenyl)-5-methyl-4-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-oxazole
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]ethyl]methylamine
2-{8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-4-carboxamide
2-amino-N-[4-(1-benzothiophen-7-yl)-2-fluorophenyl]acetamide
N-[1-(1-cyclobutanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxy-2-phenylacetamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinolin-6-ylmethyl)benzamide
3-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-N-methylpyrrolidine-3-carboxamide
8-(butan-2-yl)-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(methylsulfanyl)-N-(oxolan-2-ylmethyl)acetamide
1-(5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
4-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
6-[(4-benzylpiperidin-1-yl)methyl]-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
6-methyl-4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[1-(4-fluorophenyl)propan-2-yl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
N-(2-ethyl-1,3-dihydroxypropan-2-yl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
methyl 3-(3-fluorobenzamido)-6-[(2-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
5-(3-fluoro-4-methoxyphenyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2,4-triazin-3-amine
2-{[2-(2,4-difluorophenyl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
5-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1,2-oxazole
1-(2,4-dichlorophenyl)-3-(2-methoxyethyl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
4-(4-methylphenoxy)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
methyl 4-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-pyrazole-3-carboxylate
N'-(3-chloro-2-methylphenyl)-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanediamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(4-phenylpiperidin-1-yl)acetamide
4-{[5-(2,4-difluoro-3-methoxyphenyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
2-[5-(2-methyl-1,3-oxazol-4-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
dimethyl({2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-1-(thiophen-2-yl)ethyl})amine
N-(2-methoxyethyl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
5-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-N-(2,2-difluoroethyl)benzene-1-sulfonamide
(2S,4R)-1-cyclobutanecarbonyl-4-(4-ethenylbenzamido)-N-ethylpyrrolidine-2-carboxamide
methyl 1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-pyrazole-3-carboxylate
(1R,5S)-3-{[4-(2-methylphenyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-6-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
(3S,4R)-1-(2-carboxyethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)oxane-4-carboxamide
2-(3-fluoro-4-methylphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(2-methyl-1,3-benzothiazol-6-yl)-1H-indazole-3-carboxamide
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]propanamide
5-[2-(benzylamino)ethyl]-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)pyrrolidin-2-one
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[3-(trifluoromethyl)phenyl]methyl}amine
7-(1-benzothiophene-2-carbonyl)-2-propyl-2,7-diazaspiro[4.5]decane
2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}ethan-1-one
1-{[5-(7-fluoro-4-methylquinolin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea