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N-cyclohexyl-N-(pyridin-4-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3,5-dichloro-2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
[3-({1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[(2,3-dimethyl-1H-indol-7-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
methyl (1R,3R,3aR,6aS)-1-benzyl-5-methyl-3-(oxan-4-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
5-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)-2-(2-methoxyethyl)pyrimidine
(4aR,7aS)-1-ethyl-4-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-(3-hydroxy-3-methylbutyl)benzoyl]-3-(2-hydroxyethyl)piperazin-2-one
2-[3-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)phenoxy]ethan-1-ol
1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-hydroxyethan-1-one
7-(2-methoxyethyl)-2-(4,7,8-trimethylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(1R,3R,5S)-8-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-8-azabicyclo[3.2.1]octan-3-ol
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
2-({[4-(1H-pyrazol-1-yl)phenyl]methyl}(thiophen-3-ylmethyl)amino)butan-1-ol
4-{[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}-2,6-dimethoxyphenol
1-methyl-8-{[4-(methylsulfanyl)phenyl]carbamoyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-({1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}sulfonyl)benzonitrile
4-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-1,2-dihydroquinolin-2-one
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-2-one
2-[4-({[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)phenyl]-N-cyclopropylacetamide
N-{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}thian-4-amine
1-[(4-chlorophenyl)methyl]-N-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-1,2,3-triazole-4-carboxamide
6-methoxy-1-methyl-N-(3-{[(2-methylphenyl)methyl]sulfanyl}propyl)-1H-indole-2-carboxamide
2-(3-hydroxypropyl)-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-({[7-chloro-2-(2-phenylethoxy)quinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
1'-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[3-oxo-9-(1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(propan-2-yloxy)ethan-1-one
2-{2-[methyl(oxan-2-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-[(1R,3R)-3-aminocyclopentyl]-5,7-dimethyl-2,1,3-benzoxadiazole-4-sulfonamide
1-(propan-2-yl)-N-[2-(pyrazin-2-yl)ethyl]piperidine-4-carboxamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
2-benzyl-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,3-thiazole-4-carboxamide
3-(piperidin-3-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
2-(dimethylamino)-N-[3-(1H-imidazol-1-yl)propyl]-4-methylpyrimidine-5-carboxamide
5-ethyl-3-{2-[2-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
5-(4-acetylphenoxymethyl)-N-[(4-fluorophenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
7-(1-benzothiophen-3-yl)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(oxan-4-ylmethyl)-3-propylpiperidine-3-carboxylic acid
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-methyl-5-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-[(3,4-difluorophenyl)methyl]-8-(pyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-({3-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-3-carboxamide
1-cyclohexanecarbonyl-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-(2H-1,3-benzodioxol-5-yl)-N-[(1-propylpyrrolidin-3-yl)methyl]piperidin-4-amine
2-(ethylamino)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-5-carboxamide