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2-[2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)ethoxy]ethan-1-ol
(3S)-1-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-ol
8-(6-chloropyridazin-3-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[(2R,4R,6S)-2-(4-chlorophenyl)-6-(1-methyl-1H-1,2,3-benzotriazol-5-yl)oxan-4-yl]acetamide
5-{4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}-1H-imidazol-2-amine
N-[2-(benzyloxy)ethyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(1-{6-[3-(aminomethyl)phenyl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
4-ethyl-1-methyl-3-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{1-[(8-methoxyquinolin-2-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
N-ethyl-2,3-difluoro-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}benzamide
N-[(3R,5S)-1-cyclopentanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
2-benzyl-8-(2,3-dihydro-1H-indene-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]propane-1,2-diol
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-[6-methyl-2-(methylamino)pyrimidin-4-yl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-[3-(4-fluorophenoxy)azetidin-1-yl]ethan-1-one
1-(1-{1-[2-(azepan-1-ylmethyl)-2-methylpropyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N,6,6-trimethyl-5-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]thiomorpholine-3-carboxamide
N-[(3-methoxy-2-propoxyphenyl)methyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(prop-2-en-1-yl)pyrimidin-2-amine
2-methoxy-4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidin-3-ol
1-[(4-fluorophenyl)methyl]-4-[4-(piperidin-3-yl)benzoyl]piperazine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
8-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-[2-(dimethylamino)-4-{[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-ethyl-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-1H-pyrazole-4-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[1-(hydroxymethyl)cyclopentyl]acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
(2S)-2-amino-3-cyclohexyl-N-[1-(methoxymethyl)cyclopentyl]propanamide
2-(3-methoxyphenyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methylpropyl)piperidine
1-{[3-(furan-2-yl)phenyl]methyl}-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
3-cyclohexyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2-hydroxyphenyl)ethan-1-one
6-ethyl-2-oxo-N-(pyridin-4-ylmethyl)-1,2-dihydropyridine-4-carboxamide
3-(3,4-difluorophenyl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]propanamide
1-ethyl-3-methyl-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}-1H-pyrazole-5-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-[1-methyl-4-(pyridin-3-ylmethyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]-3-phenylpropan-1-one
4-{1-cyclohexyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazol-3-yl}pyridine
3-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-(2-methyl-5-sulfamoylphenyl)urea
5-(4-benzylpiperidin-1-yl)-1-ethyl-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-cyclopentanecarbonyl-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
(1R,5S)-3-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-(cyclohex-1-en-1-ylmethyl)acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-methylthiophene-2-carboxamide