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2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-(1-ethylpiperidin-4-yl)acetamide
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]oxolane-2-carboxamide
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-N,2,6-trimethylpyrimidine-4-carboxamide
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methoxypiperidine
8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-N-methyl-2-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2-dihydropyridine-4-carboxamide
N-butyl-N,5-dimethyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
[(3-fluorophenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
N-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}aniline
2-({2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
3-(2,4-dimethoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
2-methyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]butanamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
N-[2-(cyclohexylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,5R)-6-(5-ethylthiophene-3-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-N-[(2-methylphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-dimethyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
(2-{2-[1-(1-benzothiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-1'-(2,2,3,3-tetramethylcyclopropanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-cyclohexyl-4-(2,2-diethylcyclopropanecarbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
[(3R,4R)-1-{[3-(2-aminoethyl)phenyl]methyl}-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
1-{2-[(4-acetylphenyl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-methoxypropan-1-one
2-ethoxy-1-[4-(3-methyl-3-phenylpiperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-4-(piperidin-1-yl)benzamide
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-[4-(2-methoxybenzoyl)piperazin-1-yl]ethan-1-one
3-(furan-2-yl)-2-[2-(thiophen-3-yl)-1H-imidazol-1-yl]propanoic acid
10-methoxy-5-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-(3,3-dimethylpyrrolidine-1-carbonyl)-7-fluoro-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
(1S,5R)-6-[(5-propylfuran-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(methylamino)pyridine-4-carboxamide
1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]acetamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)propanamide
N-({1-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}methyl)acetamide
N-(3,5-dimethoxyphenyl)-2-[(oxolan-2-ylmethyl)amino]acetamide
3-(5-{1-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-1,2,3-triazol-4-yl}thiophen-3-yl)prop-2-yn-1-ol
2-{2-[4-(1H-indol-4-ylmethyl)piperazin-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-{1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-yl}acetamide
1-{3-[(3-hydroxyazetidin-1-yl)sulfonyl]benzoyl}piperidine-3-carbonitrile
(2R)-2-amino-3-(4-chlorophenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
7-(propan-2-yl)-2-[4-(trifluoromethyl)pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-[(1,1-diphenylpropan-2-yl)amino]-3-methylbutan-1-ol
N,N-dimethyl-4-{[2-(quinolin-2-yl)-1H-imidazol-1-yl]methyl}oxan-4-amine
N-[4-({[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]amino}methyl)phenyl]acetamide