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1-{1-[(3-methoxyphenyl)methyl]-5-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3,4-dimethoxyphenyl)methyl]methylamine
N-methyl-2-[4-(5-{[(2-methylphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]acetamide
N-{[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}-2-methoxyacetamide
1-[(4aR,8aS)-6-(2-phenylethyl)-decahydro-1,6-naphthyridin-1-yl]-2-(4-acetylphenoxy)ethan-1-one
3-[(4-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-1H-1,2,3-triazol-1-yl)methyl]piperidine
2-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-N-methyl-N-phenylacetamide
N-methyl-3-(1-methyl-1H-pyrazol-4-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
ethyl 4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
N-(adamantan-2-ylmethyl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]acetamide
2-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-chloro-5-acetamido-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
2-[4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
3,5-dimethyl-1-(4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}phenyl)-1H-pyrazole
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
5-[(6-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-methoxy-2-methylpropan-1-one
3-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
N-(1-methylpiperidin-4-yl)-5-phenyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-[2-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
1-(5-chloropyridin-2-yl)-4-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperazine
N-[4-(1H-indol-2-yl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-cyclohexylpiperazine
1-({1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}methyl)pyrrolidin-2-one
3-[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{6-hydroxy-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepan-1-yl}-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
2-[5-(8-chloroquinolin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
2-{4-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-1H-pyrazol-1-yl}-N-methylacetamide
3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidine-1-carboxamide
6-[({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)methyl]pyrimidin-4-ol
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)pent-4-enamide
1-{[4-(difluoromethoxy)phenyl]methyl}-2-(methoxymethyl)piperidine
3-(2-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
3-(4-chloro-2-methylbenzoyl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
4-(4-fluorophenyl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1,2,3,6-tetrahydropyridine
2,8-dimethyl-N-[1-(pyridin-3-yl)propan-2-yl]quinoline-4-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-N-methyl-1,3-thiazol-2-amine
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
methyl(2-phenylethyl)({3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,2-oxazol-5-yl}methyl)amine
1-(diethylamino)-3-(2-methoxy-4-{[(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
methyl 1-benzyl-3-cyclopropaneamido-5-{[(3,4,5-trimethoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methyl-1H-1,3-benzodiazol-2-yl)methanol
1-(2-methoxyethyl)-8-(propan-2-yl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide