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2-{1-[6-(2-chlorophenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-2-yl]-N-methylformamido}propanamide
(1R,5R)-6-(cyclobutylmethyl)-3-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-(3-aminoazepan-1-yl)-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
3-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-(propan-2-yl)-1,2,4-oxadiazole
3-{2-[3-(2-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
2-ethyl-7-methoxy-4-[(4-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,8aR)-6-(5-fluoropyrimidin-2-yl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
3-methyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]but-2-enamide
2-butyl-4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
2-(4-hydroxyphenyl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
2-amino-3-ethyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-{[({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)amino]methyl}pyrrolidin-2-yl]methanol
2-methyl-8-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,3S)-3-(2-aminoethoxy)-7-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-7-azaspiro[3.5]nonan-1-ol
N-cyclopropyl-2-methyl-6-(piperidin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
2-{5-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-(cyclohex-3-en-1-ylmethyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
6-[(4-benzoylpiperidin-1-yl)methyl]-1,4-oxazepan-6-ol
4-(4-ethyl-5-methylpyrimidin-2-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(cyclohex-1-en-1-ylmethyl)-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
8-fluoro-3-(2-hydroxypropyl)-3,4-dihydroquinazolin-4-one
N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1,3-benzothiazole-2-carboxamide
N-(1-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
9-[(3-fluorophenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[5-(morpholin-4-yl)pentyl]acetamide
6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{2-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-1H-imidazole
2-(methylsulfanyl)-4-(4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)pyrimidine
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-(1H-indol-5-ylmethyl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]ethan-1-one
1-cyclopentanecarbonyl-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
[(5-chlorofuran-2-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
4-amino-N-({1-[(3-methylphenyl)methyl]piperidin-3-yl}methyl)pyridine-2-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-4-oxo-2-propyl-1,4-dihydropyridine-3-carboxamide
N-[4-(3-fluorophenyl)phenyl]-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
5-(azepane-1-carbonyl)-1-[2-(3-fluorophenyl)ethyl]piperidin-2-one
3-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
2-[(4-methoxyphenyl)methyl]-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)morpholine
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(4-hydroxyphenyl)propanamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]furan-3-carboxamide
1-(3-oxo-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propyl)azepan-2-one
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[2-(1H-pyrazol-4-yl)ethyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carboxamide
9-benzoyl-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
N,1,3-trimethyl-N-(2-phenyl-1-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}ethyl)-1H-pyrazole-5-carboxamide