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N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-[(4-chlorophenyl)methyl]-4-hydroxy-N-propyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(3R,4R)-3,4-dimethyl-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-3-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-4-carboxamide
4-{[3-(3-methoxyphenoxymethyl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
3-[(cyclopentylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-(1-hydroxypropan-2-yl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-(2-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
4-{[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
2,3,5-trimethyl-6-[6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]pyrazine
3-methoxy-1-(2-oxo-2-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}ethyl)-1,2-dihydropyridin-2-one
1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperidine-3-carboxamide
3-[4-(2-methanesulfonylethyl)piperazin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-(cyclopropylmethyl)-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
9-methoxy-3-{[4-(pyrrolidin-1-yl)phenyl]methyl}-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
5-[2-(benzylamino)ethyl]-1-[3-(pyridin-4-yl)propyl]pyrrolidin-2-one
5-fluoro-N-methyl-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
3,4,5-trimethoxy-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
N5-cycloheptyl-1-cyclopropyl-N3-methyl-N3-[2-(4-methylphenoxy)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
4-[3-(4-fluorophenoxy)propyl]-1-(3-methoxyphenyl)piperazin-2-one
1-[(3,4-dimethoxypyridin-2-yl)methyl]azepan-3-amine
7-(3-chlorophenyl)-4-(morpholine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-(2-methoxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-(2-methyl-1-benzofuran-5-yl)thiomorpholine-4-carboxamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-(3-methylphenoxy)azetidine-1-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
N-[(4-fluorophenyl)methyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
N-(furan-2-ylmethyl)-4-methyl-5-(1-phenyl-1H-pyrazol-3-yl)-1,3-thiazol-2-amine
[(4-fluorophenyl)methyl][(6-methoxypyridin-3-yl)methyl](pyridin-4-ylmethyl)amine
3-(2-methoxy-5-methylphenyl)-5-(trifluoromethyl)-1H-1,2,4-triazole
(1S,5R)-3-benzyl-6-(ethanesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(oxolan-3-yl)amino]pyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-5-(oxan-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-propyl-4-[({[1-(pyrrolidin-1-yl)cyclopentyl]methyl}carbamoyl)amino]benzamide
1-[4-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-(3,4-dimethylphenyl)-1-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(1,1,2,2-tetrafluoroethoxy)benzamide
5-(4-fluorophenyl)-N-[3-(morpholin-4-yl)propyl]-1,2,4-triazin-3-amine
6-(4-methylpiperidin-1-yl)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
1'-(5-methoxy-4-oxo-1,4-dihydropyridine-2-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N4-(1-benzoylpiperidin-3-yl)-6-ethyl-5-methylpyrimidine-2,4-diamine
2-(hydroxymethyl)-N-{2-[methyl(phenyl)amino]propyl}-1H-1,3-benzodiazole-5-carboxamide
2-{4-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-2-oxopiperazin-1-yl}benzonitrile